Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 11043
LigandPNGBDBM587720(2-[({8-[(2-methylbiphenyl-3-yl)amino]-1,7-naphthyr...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
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Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587739(2-cyclohex-1-en-1-yl-6-[(3-{[(2-hydroxyethyl)amino...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587723(1-({8-[(2-methylbiphenyl-3-yl)amino]-1,7-naphthyri...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587738(3-[(3-{[(2-hydroxyethyl)amino]methyl}-1,7-naphthyr...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587737(2-[({8-[(3-cyclohex-1-en-1-yl-2-methylphenyl)amino...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587736(2-{[(8-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-me...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587735(2-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-[(3-{[(2-hy...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587728(2-[({4-methoxy-8-[(2-methylbiphenyl-3-yl)amino]-1,...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587730(2-{[(8-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-me...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587732(2-[({5-[(2-methylbiphenyl-3-yl)amino]pyrido[3,4-b]...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587740(2-cyclohexyl-6-[(3-{[(2-hydroxyethyl)amino]methyl}...)
Affinity DataIC50: 55nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM50542976(CHEMBL4636606 | US11535615, Example 1)
Affinity DataIC50: 55nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587734((2S)-1-({5-[(2-methylbiphenyl-3-yl)amino]pyrido[3,...)
Affinity DataIC50: 55nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587731(1-[(8-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-met...)
Affinity DataIC50: 55nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587729(1-({4-chloro-8-[(2-methylbiphenyl-3-yl)amino]-1,7-...)
Affinity DataIC50: 55nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587727(2-[({4-chloro-8-[(2-methylbiphenyl-3-yl)amino]-1,7...)
Affinity DataIC50: 55nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587726(1-({8-[(2-methylbiphenyl-3-yl)amino]quinolin-4-yl}...)
Affinity DataIC50: 55nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587725(2-[({8-[(2-methylbiphenyl-3-yl)amino]quinolin-4-yl...)
Affinity DataIC50: 55nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587724(2-[({8-[(2-methylbiphenyl-3-yl)amino]-1,7-naphthyr...)
Affinity DataIC50: 55nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587722(1-({4-[(2-methylbiphenyl-3-yl)amino]pyrido[3,2-d]p...)
Affinity DataIC50: 55nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
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LigandPNGBDBM587721(1-({8-[(2-methylbiphenyl-3-yl)amino]-1,7-naphthyri...)
Affinity DataIC50: 55nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/20/2023
Entry Details
Go to US Patent