Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 10818
LigandPNGBDBM50502718(CHEMBL4464675 | US11440915, Example 12)
Affinity DataEC50:  49nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
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LigandPNGBDBM571407(US11440915, Example 22 | (9R)-N-[4-(4-methylimidaz...)
Affinity DataEC50:  27nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
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LigandPNGBDBM571406(US11440915, Example 21 | (9R)-N-[4-(4-methylimidaz...)
Affinity DataEC50:  43nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
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LigandPNGBDBM571405(US11440915, Example 20 | (9R)-N-[3-(4-methylimidaz...)
Affinity DataEC50:  10nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
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LigandPNGBDBM571404(US11440915, Example 19 | (9R)-N-[3-(4-methylimidaz...)
Affinity DataEC50:  14nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM571403(US11440915, Example 18 | (9R)-9-(2-fluorophenyl)-N...)
Affinity DataEC50:  62nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM571402(US11440915, Example 17 | (9R)-9-(2-fluorophenyl)-N...)
Affinity DataEC50:  56nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM571401(US11440915, Example 16 | (9R)-9-(2-fluorophenyl)-N...)
Affinity DataEC50:  19nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM571400(US11440915, Example 15 | (9R)-9-(2-fluorophenyl)-N...)
Affinity DataEC50:  38nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502722(CHEMBL4522681 | US11440915, Example 14)
Affinity DataEC50:  27nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502717(CHEMBL4461898 | US11440915, Example 13)
Affinity DataEC50:  44nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502710(CHEMBL4520800 | US11440915, Example 1)
Affinity DataEC50:  15nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502716(CHEMBL4576494 | US11440915, Example 11)
Affinity DataEC50:  39nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502715(CHEMBL4567728 | US11440915, Example 10)
Affinity DataEC50:  14nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502721(CHEMBL4435639 | US11440915, Example 9)
Affinity DataEC50:  8nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502709(CHEMBL4538936 | US11440915, Example 8)
Affinity DataEC50:  14nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502714(CHEMBL4470732 | US11440915, Example 7)
Affinity DataEC50:  15nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502713(CHEMBL4468874 | US11440915, Example 6)
Affinity DataEC50:  23nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502712(CHEMBL4439419 | US11440915, Example 5)
Affinity DataEC50:  26nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502720(CHEMBL4474921 | US11440915, Example 4)
Affinity DataEC50:  31nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502711(CHEMBL4515522 | US11440915, Example 3)
Affinity DataEC50:  25nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
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Date in BDB:
11/19/2022
Entry Details
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LigandPNGBDBM50502719(CHEMBL4475670 | US11440915, Example 2)
Affinity DataEC50:  16nMAssay Description:Human neuroglioma H4 cells overexpressing human APP695 with the Swedish double mutation (K595N/M596L) were plated at 30,000 cells/well/100 μl in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
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