Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 10740
LigandPNGBDBM50318482(CHEMBL470670 | l-menthol | (-)-menthol | MENTHOL |...)
Affinity DataEC50:  3.80E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
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LigandPNGBDBM562648(US11406649, Code DIPA-1-5 | 1-Di(isopropyl)- phosp...)
Affinity DataEC50:  5.60E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
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LigandPNGBDBM562695(US11406649, Code DIPA-1-6 | 1-Di(isopropyl)- phosp...)
Affinity DataEC50:  2.40E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
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LigandPNGBDBM562697(US11406649, Code DIPA-1-7 | 1-Di(isopropyl)- phosp...)
Affinity DataEC50:  700nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
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LigandPNGBDBM562698(US11406649, Code DIPA-1-8 | 1-Di(isopropyl)- phosp...)
Affinity DataEC50:  700nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
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LigandPNGBDBM562746(US11406649, Code DIPA-1-9 | 1-Diispropyl- phosphin...)
Affinity DataEC50:  900nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
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PDB3D3D Structure (crystal)
LigandPNGBDBM562747(US11406649, Code DAPA-2-4 | 1-Di(sec-butyl)- phosp...)
Affinity DataEC50:  1.45E+4nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
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LigandPNGBDBM562748(US11406649, Code DAPA-2-5 | 1-Di(sec-butyl)-phosph...)
Affinity DataEC50:  1.70E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
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LigandPNGBDBM562749(US11406649, Code DAPA-2-6 | 1-Di(sec-butyl)- phosp...)
Affinity DataEC50:  800nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
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LigandPNGBDBM562750(US11406649, Code DAPA-2-7 | 1-Di(sec-butyl)- phosp...)
Affinity DataEC50:  1.10E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
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LigandPNGBDBM562751(US11406649, Code DAPA-2-8 | 1-Di(sec-butyl)- phosp...)
Affinity DataEC50:  1.30E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
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LigandPNGBDBM562752(US11406649, Code DAPA-3-1 | 1-di(iso-butyl) phosph...)
Affinity DataEC50:  2.40E+4nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
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LigandPNGBDBM562753(US11406649, Code DAPA-3-2 | 1-Di(sec-butyl) phosph...)
Affinity DataEC50:  4.20E+3nMAssay Description:In the first set of data, the potency and in vitro effects of test compounds were evaluated on cloned hTRPM8 channel (encoded by the human TRPM8 gene...More data for this Ligand-Target Pair
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Date in BDB:
10/28/2022
Entry Details
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