Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 10722
TargetCYP1A(Human)
The General Hospital

US Patent
LigandPNGBDBM50051349(4-Methoxy-7-methyl-furo[3,2-g]chromen-5-one | CHEM...)
Affinity DataIC50: 240nMAssay Description:The ability of the tested compounds to inhibit a panel of CYP enzymes in vitro was assessed using a series of human liver microsome assays. Half-maxi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2022
Entry Details
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TargetCYP1A(Human)
The General Hospital

US Patent
LigandPNGBDBM562067(US11396516, Example 2)
Affinity DataIC50: 1.60E+3nMAssay Description:The ability of the tested compounds to inhibit a panel of CYP enzymes in vitro was assessed using a series of human liver microsome assays. Half-maxi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2022
Entry Details
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TargetCytochrome P450 2D6(Human)
The General Hospital

US Patent
LigandPNGBDBM562067(US11396516, Example 2)
Affinity DataIC50: 2.00E+3nMAssay Description:The ability of the tested compounds to inhibit a panel of CYP enzymes in vitro was assessed using a series of human liver microsome assays. Half-maxi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2022
Entry Details
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TargetCytochrome P450 3A43(Human)
The General Hospital

US Patent
LigandPNGBDBM562067(US11396516, Example 2)
Affinity DataIC50: 9.30E+3nMAssay Description:The ability of the tested compounds to inhibit a panel of CYP enzymes in vitro was assessed using a series of human liver microsome assays. Half-maxi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2022
Entry Details
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TargetCytochrome P450 2C19(Human)
The General Hospital

US Patent
LigandPNGBDBM562067(US11396516, Example 2)
Affinity DataIC50: 1.20E+4nMAssay Description:The ability of the tested compounds to inhibit a panel of CYP enzymes in vitro was assessed using a series of human liver microsome assays. Half-maxi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2022
Entry Details
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TargetCytochrome P450 2B6(Human)
The General Hospital

US Patent
LigandPNGBDBM562067(US11396516, Example 2)
Affinity DataIC50: 8.80E+4nMAssay Description:The ability of the tested compounds to inhibit a panel of CYP enzymes in vitro was assessed using a series of human liver microsome assays. Half-maxi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2022
Entry Details
Go to US Patent