Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 10617
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Pittsburgh

US Patent
LigandPNGBDBM554543(US11339122, Compound 14)
Affinity DataKi:  470nMAssay Description:Binding studies with [3H]RTX were carried out as follows. The binding assay mixtures were prepared in 1.5 ml centrifuge tubes and consisted of a fixe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2022
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Pittsburgh

US Patent
LigandPNGBDBM554544(US11339122, Compound 15)
Affinity DataKi:  490nMAssay Description:Binding studies with [3H]RTX were carried out as follows. The binding assay mixtures were prepared in 1.5 ml centrifuge tubes and consisted of a fixe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2022
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Pittsburgh

US Patent
LigandPNGBDBM554545(US11339122, Compound 16)
Affinity DataKi:  560nMAssay Description:Binding studies with [3H]RTX were carried out as follows. The binding assay mixtures were prepared in 1.5 ml centrifuge tubes and consisted of a fixe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2022
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Pittsburgh

US Patent
LigandPNGBDBM554546(US11339122, Compound 17)
Affinity DataKi:  2.15E+3nMAssay Description:Binding studies with [3H]RTX were carried out as follows. The binding assay mixtures were prepared in 1.5 ml centrifuge tubes and consisted of a fixe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2022
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Pittsburgh

US Patent
LigandPNGBDBM554537(US11339122, Compound 1)
Affinity DataKi:  2.57E+3nMAssay Description:Binding studies with [3H]RTX were carried out as follows. The binding assay mixtures were prepared in 1.5 ml centrifuge tubes and consisted of a fixe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2022
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Pittsburgh

US Patent
LigandPNGBDBM46760(cid_306328 | ethyl 4-[(4-fluorophenyl)carbamoylami...)
Affinity DataKi:  2.84E+3nMAssay Description:Binding studies with [3H]RTX were carried out as follows. The binding assay mixtures were prepared in 1.5 ml centrifuge tubes and consisted of a fixe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2022
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Pittsburgh

US Patent
LigandPNGBDBM554542(US11339122, Compound 13)
Affinity DataKi:  3.70E+3nMAssay Description:Binding studies with [3H]RTX were carried out as follows. The binding assay mixtures were prepared in 1.5 ml centrifuge tubes and consisted of a fixe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2022
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Pittsburgh

US Patent
LigandPNGBDBM554541(US11339122, Compound 11)
Affinity DataKi:  3.70E+3nMAssay Description:Binding studies with [3H]RTX were carried out as follows. The binding assay mixtures were prepared in 1.5 ml centrifuge tubes and consisted of a fixe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2022
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Pittsburgh

US Patent
LigandPNGBDBM554538(US11339122, Compound 2)
Affinity DataKi:  4.52E+3nMAssay Description:Binding studies with [3H]RTX were carried out as follows. The binding assay mixtures were prepared in 1.5 ml centrifuge tubes and consisted of a fixe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2022
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Pittsburgh

US Patent
LigandPNGBDBM554547(US11339122, Compound 18)
Affinity DataKi:  7.00E+3nMAssay Description:Binding studies with [3H]RTX were carried out as follows. The binding assay mixtures were prepared in 1.5 ml centrifuge tubes and consisted of a fixe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2022
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Pittsburgh

US Patent
LigandPNGBDBM554539(US11339122, Compound 4)
Affinity DataKi:  1.17E+4nMAssay Description:Binding studies with [3H]RTX were carried out as follows. The binding assay mixtures were prepared in 1.5 ml centrifuge tubes and consisted of a fixe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2022
Entry Details
US Patent