Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 10310
TargetTyrosine-protein kinase BTK(Human)
Shenzhen Targetrx

US Patent
LigandPNGBDBM526931((S)-1-(3-(4-amino-5-(4-phenoxyphenyl)-5H-pyrrolo[3...)
Affinity DataIC50: 1nMAssay Description:BTK (Invitrogen, catalog number: PR5442A), HTRF-TK kit (Cisbio, catalog number: 62TK0PEC), MgCl2 (SIGMA, catalog number: 63020-1L), ATP (Sigma, catal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetTyrosine-protein kinase BTK(Human)
Shenzhen Targetrx

US Patent
LigandPNGBDBM526932((R)-1-(3-(4-amino-5-(4-phenoxyphenyl)-5H-pyrrolo[3...)
Affinity DataIC50: 1nMAssay Description:BTK (Invitrogen, catalog number: PR5442A), HTRF-TK kit (Cisbio, catalog number: 62TK0PEC), MgCl2 (SIGMA, catalog number: 63020-1L), ATP (Sigma, catal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Shenzhen Targetrx

US Patent
LigandPNGBDBM526933((R)-1-(3-(7-amino-1-(4-phenoxyphenyl)-1H-pyrazolo[...)
Affinity DataIC50: 1nMAssay Description:BTK (Invitrogen, catalog number: PR5442A), HTRF-TK kit (Cisbio, catalog number: 62TK0PEC), MgCl2 (SIGMA, catalog number: 63020-1L), ATP (Sigma, catal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Shenzhen Targetrx

US Patent
LigandPNGBDBM526934((S)-1-(3-(7-amino-1-(4-phenoxyphenyl)-1H-pyrazolo[...)
Affinity DataIC50: 1nMAssay Description:BTK (Invitrogen, catalog number: PR5442A), HTRF-TK kit (Cisbio, catalog number: 62TK0PEC), MgCl2 (SIGMA, catalog number: 63020-1L), ATP (Sigma, catal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Shenzhen Targetrx

US Patent
LigandPNGBDBM526935((S)-1-(3-(8-amino-1-(4-phenoxyphenyl)-1H-pyrazolo[...)
Affinity DataIC50: 1nMAssay Description:BTK (Invitrogen, catalog number: PR5442A), HTRF-TK kit (Cisbio, catalog number: 62TK0PEC), MgCl2 (SIGMA, catalog number: 63020-1L), ATP (Sigma, catal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Shenzhen Targetrx

US Patent
LigandPNGBDBM50357312(IBRUTINIB | US9181263, 1 | US9108973, Ref 1 | US92...)
Affinity DataIC50: 1nMAssay Description:BTK (Invitrogen, catalog number: PR5442A), HTRF-TK kit (Cisbio, catalog number: 62TK0PEC), MgCl2 (SIGMA, catalog number: 63020-1L), ATP (Sigma, catal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
Go to US Patent