Compile Data Set for Download or QSAR
Report error Found 90 Enz. Inhib. hit(s) with all data for entry = 10329
LigandPNGBDBM528351(US11180503, Example 9 | 9-([1,1'- Bi(cyclopropan)]...)
Affinity DataIC50: 0.214nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
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LigandPNGBDBM528352(US11180503, Example 10 | 9-([1,1'-bi(cyclopropan)]...)
Affinity DataIC50: 0.260nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528349(US11180503, Example 7 | 9-([1,1'- Bi(cyclopropan)]...)
Affinity DataIC50: 0.343nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528331(US11180503, Example 1 | 9-([1,1'-bi(cyclopropan)]-...)
Affinity DataIC50: 0.366nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528352(US11180503, Example 10 | 9-([1,1'-bi(cyclopropan)]...)
Affinity DataIC50: 0.396nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528349(US11180503, Example 7 | 9-([1,1'- Bi(cyclopropan)]...)
Affinity DataIC50: 0.400nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528331(US11180503, Example 1 | 9-([1,1'-bi(cyclopropan)]-...)
Affinity DataIC50: 0.406nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528351(US11180503, Example 9 | 9-([1,1'- Bi(cyclopropan)]...)
Affinity DataIC50: 0.419nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528355(US11180503, Example 13 | 9-([1,1'-bi(cyclopropan)]...)
Affinity DataIC50: 0.816nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528353(US11180503, Example 11 | 9-([1,1'-bi(cyclopropan)]...)
Affinity DataIC50: 0.928nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528353(US11180503, Example 11 | 9-([1,1'-bi(cyclopropan)]...)
Affinity DataIC50: 0.996nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528355(US11180503, Example 13 | 9-([1,1'-bi(cyclopropan)]...)
Affinity DataIC50: 1.13nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528334(US11180503, Example 4 | rac-9-([1,1''- Bi(cyclopro...)
Affinity DataIC50: 1.49nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528350(US11180503, Example 8 | 5-butyl-3-ethyl-9-(1-methy...)
Affinity DataIC50: 2nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528334(US11180503, Example 4 | rac-9-([1,1''- Bi(cyclopro...)
Affinity DataIC50: 2nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528349(US11180503, Example 7 | 9-([1,1'- Bi(cyclopropan)]...)
Affinity DataIC50: 2nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528352(US11180503, Example 10 | 9-([1,1'-bi(cyclopropan)]...)
Affinity DataIC50: 2nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528348(US11180503, Example 6 | 5-butyl-3-methyl-9-(1-meth...)
Affinity DataIC50: 2nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528351(US11180503, Example 9 | 9-([1,1'- Bi(cyclopropan)]...)
Affinity DataIC50: 2nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528353(US11180503, Example 11 | 9-([1,1'-bi(cyclopropan)]...)
Affinity DataIC50: 2nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528354(US11180503, Example 12 | 5-Butyl-3- (hydroxymethyl...)
Affinity DataIC50: 2nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528334(US11180503, Example 4 | rac-9-([1,1''- Bi(cyclopro...)
Affinity DataIC50: 2nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528333(US11180503, Example 3 | 9-([1,1'- Bi(cyclopropan)]...)
Affinity DataIC50: 2nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528332(US11180503, Example 2 | 5-Butyl-3- methyl-9-(1- (t...)
Affinity DataIC50: 2nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528347(US11180503, Example 5 | 9-([1,1'-bi(cylopropan)]-1...)
Affinity DataIC50: 2.41nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528333(US11180503, Example 3 | 9-([1,1'- Bi(cyclopropan)]...)
Affinity DataIC50: 2.59nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
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LigandPNGBDBM528347(US11180503, Example 5 | 9-([1,1'-bi(cylopropan)]-1...)
Affinity DataIC50: 2.75nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528347(US11180503, Example 5 | 9-([1,1'-bi(cylopropan)]-1...)
Affinity DataIC50: 3nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528355(US11180503, Example 13 | 9-([1,1'-bi(cyclopropan)]...)
Affinity DataIC50: 3nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528333(US11180503, Example 3 | 9-([1,1'- Bi(cyclopropan)]...)
Affinity DataIC50: 3.41nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528331(US11180503, Example 1 | 9-([1,1'-bi(cyclopropan)]-...)
Affinity DataIC50: 4nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528350(US11180503, Example 8 | 5-butyl-3-ethyl-9-(1-methy...)
Affinity DataIC50: 8.01nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528332(US11180503, Example 2 | 5-Butyl-3- methyl-9-(1- (t...)
Affinity DataIC50: 8.62nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528350(US11180503, Example 8 | 5-butyl-3-ethyl-9-(1-methy...)
Affinity DataIC50: 9.34nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528348(US11180503, Example 6 | 5-butyl-3-methyl-9-(1-meth...)
Affinity DataIC50: 11.6nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528332(US11180503, Example 2 | 5-Butyl-3- methyl-9-(1- (t...)
Affinity DataIC50: 12.1nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528334(US11180503, Example 4 | rac-9-([1,1''- Bi(cyclopro...)
Affinity DataIC50: 13.9nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528334(US11180503, Example 4 | rac-9-([1,1''- Bi(cyclopro...)
Affinity DataIC50: 15.1nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528348(US11180503, Example 6 | 5-butyl-3-methyl-9-(1-meth...)
Affinity DataIC50: 15.4nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528354(US11180503, Example 12 | 5-Butyl-3- (hydroxymethyl...)
Affinity DataIC50: 17.4nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528354(US11180503, Example 12 | 5-Butyl-3- (hydroxymethyl...)
Affinity DataIC50: 23nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528334(US11180503, Example 4 | rac-9-([1,1''- Bi(cyclopro...)
Affinity DataIC50: 25.8nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528334(US11180503, Example 4 | rac-9-([1,1''- Bi(cyclopro...)
Affinity DataIC50: 26.8nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528334(US11180503, Example 4 | rac-9-([1,1''- Bi(cyclopro...)
Affinity DataIC50: 33.5nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528334(US11180503, Example 4 | rac-9-([1,1''- Bi(cyclopro...)
Affinity DataIC50: 40.1nMAssay Description:PDE1B, PDE1A, and PDE1C are cloned and purified following standard protein generation procedures. The assay buffer is prepared to give a final concen...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528352(US11180503, Example 10 | 9-([1,1'-bi(cyclopropan)]...)
Affinity DataIC50: 611nMAssay Description:The following phosphodiesterase activities are measured using [3H]cGMP as reaction substrate: human PDE6A/6B. The catalytic active form of human PDE6...More data for this Ligand-Target Pair
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Date in BDB:
4/10/2022
Entry Details
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TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Human)
Eli Lilly

US Patent
LigandPNGBDBM528351(US11180503, Example 9 | 9-([1,1'- Bi(cyclopropan)]...)
Affinity DataIC50: 675nMAssay Description:The following phosphodiesterase activities are measured using [3H]cAMP as reaction substrate: human PDE3A (catalytic domain) and human PDE4D. Both en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Human)
Eli Lilly

US Patent
LigandPNGBDBM528350(US11180503, Example 8 | 5-butyl-3-ethyl-9-(1-methy...)
Affinity DataIC50: 957nMAssay Description:The following phosphodiesterase activities are measured using [3H]cAMP as reaction substrate: human PDE3A (catalytic domain) and human PDE4D. Both en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Human)
Eli Lilly

US Patent
LigandPNGBDBM528352(US11180503, Example 10 | 9-([1,1'-bi(cyclopropan)]...)
Affinity DataIC50: 972nMAssay Description:The following phosphodiesterase activities are measured using [3H]cAMP as reaction substrate: human PDE3A (catalytic domain) and human PDE4D. Both en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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LigandPNGBDBM528351(US11180503, Example 9 | 9-([1,1'- Bi(cyclopropan)]...)
Affinity DataIC50: 982nMAssay Description:The following phosphodiesterase activities are measured using [3H]cGMP as reaction substrate: human PDE6A/6B. The catalytic active form of human PDE6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2022
Entry Details
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