Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 10267
TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524042(US11136333, Compound 12a)
Affinity DataKd:  3.5nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524050(US11136333, Compound 19bbIC50)
Affinity DataKd:  0.660nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524049(US11136333, Compound 19a)
Affinity DataKd:  0.380nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524048(US11136333, Compound 12g)
Affinity DataKd:  0.910nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524047(US11136333, Compound 12f)
Affinity DataKd:  1.5nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524046(US11136333, Compound 12e)
Affinity DataKd:  1.5nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524045(US11136333, Compound 12d)
Affinity DataKd:  2.60nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524044(US11136333, Compound 12c)
Affinity DataKd:  0.400nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524043(US11136333, Compound 12b)
Affinity DataKd:  3.30nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM6568(PD-173955 | CHEMBL386051 | 6-(2,6-dichlorophenyl)-...)
Affinity DataKd:  0.580nMAssay Description:This assay is described in https://www.discoverx.com/kinase-data-sheets/abl1-nonphosphorylated.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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PDB3D3D Structure (crystal)
TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524049(US11136333, Compound 19a)
Affinity DataIC50: 1.27nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524050(US11136333, Compound 19bbIC50)
Affinity DataIC50: 2.09nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524044(US11136333, Compound 12c)
Affinity DataIC50: 2.13nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524048(US11136333, Compound 12g)
Affinity DataIC50: 3.51nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524047(US11136333, Compound 12f)
Affinity DataIC50: 15.7nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524046(US11136333, Compound 12e)
Affinity DataIC50: 16.1nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524042(US11136333, Compound 12a)
Affinity DataIC50: 17.5nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524043(US11136333, Compound 12b)
Affinity DataIC50: 18.7nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
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TargetTyrosine-protein kinase ABL1(Human)
Texas A&M University System

US Patent
LigandPNGBDBM524045(US11136333, Compound 12d)
Affinity DataIC50: 42.6nMAssay Description:IC50 against Abelson kinase ABL1 was determined by Life Technologies corporation though the Z′-LITE biochemical assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
Go to US Patent