Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 10121
TargetProstacyclin receptor(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM357269(US10214518, Compound 90 | 2-(((1s,4s)-4-((5- (ethy...)
Affinity DataEC50:  7nMAssay Description:Principle of the assay: The HTRF assay kit was purchased from Cisbio-US, Inc. (Bedford, Mass.; Catalog #62AM4PEC). The HTRF assay supported by the ki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2022
Entry Details
Go to US Patent

TargetProstacyclin receptor(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM357270(US10214518, Compound 111 | 2-(((1s,4s)-4-((5- (met...)
Affinity DataEC50:  16nMAssay Description:Principle of the assay: The HTRF assay kit was purchased from Cisbio-US, Inc. (Bedford, Mass.; Catalog #62AM4PEC). The HTRF assay supported by the ki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2022
Entry Details
Go to US Patent

TargetProstacyclin receptor(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM357271(US10214518, Compound 184 | 2-(((1s,4s)-4-((5- (cya...)
Affinity DataEC50:  11nMAssay Description:Principle of the assay: The HTRF assay kit was purchased from Cisbio-US, Inc. (Bedford, Mass.; Catalog #62AM4PEC). The HTRF assay supported by the ki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2022
Entry Details
Go to US Patent

TargetProstacyclin receptor(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM357272(US10214518, Compound 198 | 2-(((1s,4s)-4-((5-(2- h...)
Affinity DataEC50:  2nMAssay Description:Principle of the assay: The HTRF assay kit was purchased from Cisbio-US, Inc. (Bedford, Mass.; Catalog #62AM4PEC). The HTRF assay supported by the ki...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2022
Entry Details
Go to US Patent