Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 10067
TargetKetohexokinase(Human)
Regents of The University of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511679(US11083720, Compound C-1 | 4-(1-phenyl-1H-indazol-...)
Affinity DataIC50: 1.17nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2022
Entry Details
US Patent

TargetKetohexokinase(Human)
Regents of The University of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511678(US11083720, Compound C-5 | 4-(1-(m-tolyl)-1H-indaz...)
Affinity DataIC50: 280nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2022
Entry Details
US Patent

TargetKetohexokinase(Human)
Regents of The University of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511689(US11083720, Compound C-25 | N-(1-(m-tolyl)-1H-inda...)
Affinity DataIC50: 510nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2022
Entry Details
US Patent

TargetKetohexokinase(Human)
Regents of The University of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511686(US11083720, Compound C-34 | N-(azetidin-3-yl)-1-ph...)
Affinity DataIC50: 580nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2022
Entry Details
US Patent

TargetKetohexokinase(Human)
Regents of The University of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511683(US11083720, Compound C-28 | 4-(3-cyclopropyl-1-phe...)
Affinity DataIC50: 700nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2022
Entry Details
US Patent

TargetKetohexokinase(Human)
Regents of The University of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511687(US11083720, Compound C-32 | N-(piperidin-4-yl)-1-(...)
Affinity DataIC50: 790nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2022
Entry Details
US Patent

TargetKetohexokinase(Human)
Regents of The University of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511690(US11083720, Compound C-72)
Affinity DataIC50: 1.20E+3nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2022
Entry Details
US Patent

TargetKetohexokinase(Human)
Regents of The University of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511684(US11083720, Compound C-33 | N-(azetidin-3-yl)-1-(m...)
Affinity DataIC50: 2.30E+3nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2022
Entry Details
US Patent

TargetKetohexokinase(Human)
Regents of The University of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511688(US11083720, Compound C-26 | 1-phenyl-N-(piperidin-...)
Affinity DataIC50: 2.30E+3nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/23/2022
Entry Details
US Patent