Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 10007
TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
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US Patent
LigandPNGBDBM507637(US11046681, Example 165 | 1-(2,3-dihydro-1,4-benzo...)
Affinity DataIC50: 19.6nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
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US Patent
LigandPNGBDBM507626(US11046681, Example 135 | 3-[[4-hydroxy-1-[(3R,4R)...)
Affinity DataIC50: 28.7nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
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US Patent
LigandPNGBDBM507620(US11046681, Example 101 | 3-[[4-hydroxy-1-[(3R,4R)...)
Affinity DataIC50: 31.6nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
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US Patent
LigandPNGBDBM507625(US11046681, Example 130 | 7-(4-fluorophenyl)-3-[[4...)
Affinity DataIC50: 37.7nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
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US Patent
LigandPNGBDBM507635(US11046681, Example 157 | 7-(4-fluoro-3-methoxy-ph...)
Affinity DataIC50: 39.3nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
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US Patent
LigandPNGBDBM507630(US11046681, Example 143 | 7-(4-chlorophenyl)-3-[[4...)
Affinity DataIC50: 41.2nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
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US Patent
LigandPNGBDBM507634(US11046681, Example 153 | 7-(4-chlorophenyl)-3-[[4...)
Affinity DataIC50: 48.6nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507627(US11046681, Example 136 | 3-[[4-hydroxy-1-[(3R,4R)...)
Affinity DataIC50: 48.6nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507616(US11046681, Example 40 | tert-butyl (3R,4R)-4-[4-h...)
Affinity DataIC50: 49.9nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
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US Patent
LigandPNGBDBM507632(US11046681, Example 151 | 3-[[4-hydroxy-1-[(3R,4R)...)
Affinity DataIC50: 52.4nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
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US Patent
LigandPNGBDBM507621(US11046681, Example 103 | 5-[[4-hydroxy-1-[(3R,4R)...)
Affinity DataIC50: 52.9nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507629(US11046681, Example 142 | 7-(3-chlorophenyl)-3-[[4...)
Affinity DataIC50: 56.7nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507617(US11046681, Example 44 | tert-butyl (3R,4R)-4-[4-h...)
Affinity DataIC50: 61.5nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507633(US11046681, Example 152 | 7-(3-chlorophenyl)-3-[[4...)
Affinity DataIC50: 64.8nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507619(US11046681, Example 64 | tert-butyl (3R,4R)-4-[4-[...)
Affinity DataIC50: 68.7nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507618(US11046681, Example 57 | tert-butyl (3R,4R)-4-[4-[...)
Affinity DataIC50: 70.2nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507644(US11046681, Example 181 | 3-[[1-[(3R,4R)-1-acetyl-...)
Affinity DataIC50: 74.2nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507628(US11046681, Example 141 | 7-(4-fluorophenyl)-3-[[4...)
Affinity DataIC50: 74.8nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507645(US11046681, Example 184 | 3-[[1-[(3R,4R)-1-(2,2-di...)
Affinity DataIC50: 83nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507642(US11046681, Example 179 | 3-[[1-[(3R,4R)-1-acetyl-...)
Affinity DataIC50: 88.4nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507646(US11046681, Example 187 | 3-[[1-[(3R,4R)-1-(3,3-di...)
Affinity DataIC50: 88.5nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
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TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507643(US11046681, Example 180 | 3-[[1-[(3R,4R)-1-acetyl-...)
Affinity DataIC50: 89nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507641(US11046681, Example 178 | 3-[[1-[(3R,4R)-1-acetyl-...)
Affinity DataIC50: 96.1nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507638(US11046681, Example 166 | 3-[[1-[(3R,4R)-1-acetyl-...)
Affinity DataIC50: 102nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507640(US11046681, Example 177 | 3-[[4-hydroxy-1-[(3R,4R)...)
Affinity DataIC50: 103nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507636(US11046681, Example 163 | 3-[[4-hydroxy-1-[(3R,4R)...)
Affinity DataIC50: 108nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507161(tert-butyl (3R,4R)-4-[4-hydroxy-4-[(4-oxothieno[2,...)
Affinity DataIC50: 128nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507624(US11046681, Example 121 | 3-[[4-hydroxy-1-[(3R,4R)...)
Affinity DataIC50: 140nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507450(tert-butyl (3R,4R)-4-[4-hydroxy-4-[[4-oxo-7-(2-pyr...)
Affinity DataIC50: 274nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507622(US11046681, Example 104 | 3-[[4-hydroxy-1-[(3R,4R)...)
Affinity DataIC50: 394nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507631(US11046681, Example 147 | 3-[[1-[(3R,4R)-1-acetyl-...)
Affinity DataIC50: 406nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507639(US11046681, Example 169 | 5-[[1-[(3R,4R)-1,1-dimet...)
Affinity DataIC50: 860nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent

TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Les Laboratoires Servier

US Patent
LigandPNGBDBM507623(US11046681, Example 117 | 3-[[4-hydroxy-1-[(3R,4R)...)
Affinity DataIC50: 1.20E+3nMAssay Description:USP7 activity was measured using Rhodamine-110 c-terminal labelled Ubiquitin as a substrate (Viva Biosciences). Incubation with USP7 results in the r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2021
Entry Details
Go to US Patent