Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 9971
TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandPNGBDBM504316(N-(37-oxo-39-(4'-((trans)-2- | US11034991, Example...)
Affinity DataIC50: 41nMAssay Description:KDM1A inhibition assay: a multistep enzymatic reaction in which the enzyme first produces H2O2 during the demethylation of lysine 4 in a 21 AA H3K4me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2021
Entry Details
Go to US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandPNGBDBM504312(US11034991, Example 1.6 | US11034991, Example 1.1)
Affinity DataIC50: 120nMAssay Description:KDM1A inhibition assay: a multistep enzymatic reaction in which the enzyme first produces H2O2 during the demethylation of lysine 4 in a 21 AA H3K4me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2021
Entry Details
Go to US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandPNGBDBM504315(N-(37-oxo-39-(4'-((trans)-2- | US11034991, Example...)
Affinity DataIC50: 126nMAssay Description:KDM1A inhibition assay: a multistep enzymatic reaction in which the enzyme first produces H2O2 during the demethylation of lysine 4 in a 21 AA H3K4me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2021
Entry Details
Go to US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandPNGBDBM504312(US11034991, Example 1.6 | US11034991, Example 1.1)
Affinity DataIC50: 133nMAssay Description:KDM1A inhibition assay: a multistep enzymatic reaction in which the enzyme first produces H2O2 during the demethylation of lysine 4 in a 21 AA H3K4me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2021
Entry Details
Go to US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandPNGBDBM504313(N-(27-(4'-((trans)-2-(((trans)-4- | US11034991, Ex...)
Affinity DataIC50: 210nMAssay Description:KDM1A inhibition assay: a multistep enzymatic reaction in which the enzyme first produces H2O2 during the demethylation of lysine 4 in a 21 AA H3K4me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2021
Entry Details
Go to US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandPNGBDBM504314(N-(51-(4'-((trans)-2-(((trans)-4- | US11034991, Ex...)
Affinity DataIC50: 213nMAssay Description:KDM1A inhibition assay: a multistep enzymatic reaction in which the enzyme first produces H2O2 during the demethylation of lysine 4 in a 21 AA H3K4me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2021
Entry Details
Go to US Patent