Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 9777
TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM50370624(CHEMBL4169752 | US10954217, Example 00234)
Affinity DataKi:  1.70nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM50370623(CHEMBL4165863 | US10954217, Example 00237)
Affinity DataKi:  2.70nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488134(US10954217, Example Table 3.A16)
Affinity DataKi:  4nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM50370603(CHEMBL4167315 | US10954217, Example 00225)
Affinity DataKi:  4.10nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM50370571(CHEMBL4160064 | US10954217, Example 00236)
Affinity DataKi:  4.90nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM50370662(CHEMBL4161503 | US10954217, Example 00224)
Affinity DataKi:  5.90nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM50370661(CHEMBL4175187 | US10954217, Example 00253)
Affinity DataKi:  6.10nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM50370518(CHEMBL4176474 | US10954217, Example 00229)
Affinity DataKi:  8.20nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488147(US10954217, Example Table 3.A29)
Affinity DataKi:  11.7nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM50370628(CHEMBL4166276 | US10954217, Example 00262)
Affinity DataKi:  13nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488155(US10954217, Example Table 3.A37)
Affinity DataKi:  14nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM488155(US10954217, Example Table 3.A37)
Affinity DataKi:  15nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488146(US10954217, Example Table 3.A28)
Affinity DataKi:  17nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488142(US10954217, Example KTL-01-264)
Affinity DataKi:  17nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM488123(US10954217, Example Table 3.A5)
Affinity DataKi:  19nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM50370619(CHEMBL4162416 | US10954217, Example 00264)
Affinity DataKi:  19nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM50370928(CHEMBL4170703 | US10954217, Example 00255)
Affinity DataKi:  21nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM488128(US10954217, Example KTL-01-276)
Affinity DataKi:  23nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488128(US10954217, Example KTL-01-276)
Affinity DataKi:  25nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM50370625(CHEMBL4173095 | US10954217, Example 00241)
Affinity DataKi:  25nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488140(US10954217, Example KTL-01-257)
Affinity DataKi:  27nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488153(US10954217, Example Table 3.A35)
Affinity DataKi:  31nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM50370624(CHEMBL4169752 | US10954217, Example 00234)
Affinity DataKi:  33nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM488134(US10954217, Example Table 3.A16)
Affinity DataKi:  35nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM488137(US10954217, Example Table 3.A19)
Affinity DataKi:  36nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488130(US10954217, Example Table 3.A12)
Affinity DataKi:  39nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM50370518(CHEMBL4176474 | US10954217, Example 00229)
Affinity DataKi:  44nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM50370619(CHEMBL4162416 | US10954217, Example 00264)
Affinity DataKi:  48nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM50370628(CHEMBL4166276 | US10954217, Example 00262)
Affinity DataKi:  49nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488143(US10954217, Example Table 3.A25)
Affinity DataKi:  50nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM50370623(CHEMBL4165863 | US10954217, Example 00237)
Affinity DataKi:  51nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488158(US10954217, Example Table 3.A40)
Affinity DataKi:  52nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488145(US10954217, Example Table 3.A27)
Affinity DataKi:  54nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM488142(US10954217, Example KTL-01-264)
Affinity DataKi:  54nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM488160(US10954217, Example Table 3.A42)
Affinity DataKi:  56nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM50370571(CHEMBL4160064 | US10954217, Example 00236)
Affinity DataKi:  57nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM50370603(CHEMBL4167315 | US10954217, Example 00225)
Affinity DataKi:  65nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488123(US10954217, Example Table 3.A5)
Affinity DataKi:  77nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM50370661(CHEMBL4175187 | US10954217, Example 00253)
Affinity DataKi:  81nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM50370626(CHEMBL4159034 | US10954217, Example 00266)
Affinity DataKi:  83nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM488143(US10954217, Example Table 3.A25)
Affinity DataKi:  85nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488141(US10954217, Example Table 3.A23)
Affinity DataKi:  85nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488144(US10954217, Example KTL-01-184)
Affinity DataKi:  86nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488121(US10954217, Example KTL-01-121)
Affinity DataKi:  89nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM50370609(CHEMBL4177497 | US10954217, Example 00230)
Affinity DataKi:  92nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma intracellular receptor 2(Human)
University Of Texas

US Patent
LigandPNGBDBM488127(US10954217, Example KTL-01-253)
Affinity DataKi:  95nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM488146(US10954217, Example Table 3.A28)
Affinity DataKi:  97nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM488158(US10954217, Example Table 3.A40)
Affinity DataKi:  100nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM488121(US10954217, Example KTL-01-121)
Affinity DataKi:  114nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

TargetSigma non-opioid intracellular receptor 1(Human)
University Of Texas

US Patent
LigandPNGBDBM488156(US10954217, Example Table 3.A38)
Affinity DataKi:  116nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2021
Entry Details
US Patent

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