Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 9666
LigandPNGBDBM480468(N-(4-((2S,4R)-4-Amino-2-(hydroxymethyl)pyrrolidin-...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480483(N-(4-((2S,4R)-4-amino-2-(hydroxymethyl)pyrrolidin-...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480482(N-(4-((1S,4S)-2,5-Diazabicyclo[2.2.2]octan-2-yl)-2...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480481((S)—N-(4-(4,4-Difluoro-2-(hydroxymethyl)pyrro...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480480(2-(2-Fluoro-6-methoxyphenyl)-N-(2-methyl-4-(3-(pyr...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480479(2-(2-Fluoro-6-methoxyphenyl)-N-(2-methyl-4-(octahy...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480478((R)-2-(2-Fluoro-6-methoxyphenyl)-N-(2-methyl-4-(me...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480477((S)—N-(4-(3-(aminomethyl)morpholino)-2-methyl...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480476(2-(2-Fluoro-6-methoxyphenyl)-N-(2-methyl-4((1R,4R)...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480475(2-(2-Fluoro-6-methoxyphenyl)-N-(2-methyl-4-(methyl...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480474(N-(4-((2S,4S)-4-amino-2-(hydroxymethyl)pyrrolidin-...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480473(N-(4-((1R,4R)-2-Oxa-5-azabicyclo[2.2.1]heptan-5-yl...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480472(2-(2-Fluoro-6-methoxyphenyl)-N-(4((2S,4R)-2-(hydro...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480471(N-(4-((2S,4R)-4-Acetamido-2-(hydroxymethyl)pyrroli...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480470(2-(2-Fluoro-6-methoxyphenyl)-N-(4((2S,4R)-2-(hydro...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480469(2-(2-Fluoro-6-methoxyphenyl)-N-(4((2S,4R)-2-(hydro...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480452((R)—N-(4-(3-Aminopyrrolidin-1-yl)-2-methylben...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480467(N-(4-((2S,4R)-4-Amino-2-(hydroxymethyl)pyrrolidin-...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480466(N-(4-((2S,4R)-4-Amino-2-(hydroxymethyl)pyrrolidin-...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480464(N-(4-((2S,4S)-4-Amino-2-(hydroxymethyl)pyrrolidin-...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480463(N-(4-((2S,4S)-4-Amino-2-(hydroxymethyl)pyrrolidin-...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480462(N-(4-((2S,4R)-4-Amino-2-(hydroxymethyl)pyrrolidin-...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480461((S)—N-(4-(2-(Aminomethyl)pyrrolidin-1-yl)-2-(...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480460((S)—N-(4-(2-(Aminomethyl)pyrrolidin-1-yl)-2-(...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480459((S)—N-(4-(3-Aminopyrrolidin-1-yl)-7-cyano-2-m...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
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LigandPNGBDBM480458((S)—N-(4-(3-Aminopyrrolidin-1-yl)-2,7-dimethy...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
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LigandPNGBDBM480457((S)—N-(4-(3-Aminopyrrolidin-1-yl)-7-bromo-2-m...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
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LigandPNGBDBM480456((S)—N-(4-(3-Aminopyrrolidin-1-yl)-7-chloro-2-...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480455(US10899755, Example 4)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480454((R)—N-(4-(3-Aminopyrrolidin-1-yl)-2-methylben...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480453((R)—N-(4-(3-Aminopyrrolidin-1-yl)-2-methylben...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
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LigandPNGBDBM480465(N-(4-((2S,4R)-4-Amino-2-(hydroxymethyl)pyrrolidin-...)
Affinity DataKi:  300nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2021
Entry Details
Go to US Patent