Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 9626
TargetHepatocyte growth factor receptor(Human)
Lanova Medicines

US Patent
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)
Affinity DataIC50: 2.91nMAssay Description:1. Methods(1) 4 μL of prepared kinase buffer solution or 4 μL of kinase solution (100% inhibition control) were added into a 384-hole plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
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PDB3D3D Structure (crystal)
TargetHepatocyte growth factor receptor(Human)
Lanova Medicines

US Patent
LigandPNGBDBM477046(US10882853, Compound 15)
Affinity DataIC50: 6.64nMAssay Description:1. Methods(1) 4 μL of prepared kinase buffer solution or 4 μL of kinase solution (100% inhibition control) were added into a 384-hole plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
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TargetHepatocyte growth factor receptor(Human)
Lanova Medicines

US Patent
LigandPNGBDBM477041(US10882853, Compound Foretinib)
Affinity DataIC50: 7.49nMAssay Description:1. Methods(1) 4 μL of prepared kinase buffer solution or 4 μL of kinase solution (100% inhibition control) were added into a 384-hole plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
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TargetVascular endothelial growth factor receptor 2(Human)
Lanova Medicines

US Patent
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)
Affinity DataIC50: 10.6nMAssay Description:1. Methods(1) 4 μL of prepared kinase buffer solution or 4 μL of kinase solution (100% inhibition control) were added into a 384-hole plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
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TargetVascular endothelial growth factor receptor 2(Human)
Lanova Medicines

US Patent
LigandPNGBDBM477041(US10882853, Compound Foretinib)
Affinity DataIC50: 14.8nMAssay Description:1. Methods(1) 4 μL of prepared kinase buffer solution or 4 μL of kinase solution (100% inhibition control) were added into a 384-hole plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
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TargetHepatocyte growth factor receptor(Human)
Lanova Medicines

US Patent
LigandPNGBDBM477048(US10882853, Compound 33)
Affinity DataIC50: 15nMAssay Description:1. Methods(1) 4 μL of prepared kinase buffer solution or 4 μL of kinase solution (100% inhibition control) were added into a 384-hole plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
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TargetHepatocyte growth factor receptor(Human)
Lanova Medicines

US Patent
LigandPNGBDBM477044(US10882853, Compound 10)
Affinity DataIC50: 17nMAssay Description:1. Methods(1) 4 μL of prepared kinase buffer solution or 4 μL of kinase solution (100% inhibition control) were added into a 384-hole plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
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TargetHepatocyte growth factor receptor(Human)
Lanova Medicines

US Patent
LigandPNGBDBM477045(US10882853, Compound 5)
Affinity DataIC50: 20.6nMAssay Description:1. Methods(1) 4 μL of prepared kinase buffer solution or 4 μL of kinase solution (100% inhibition control) were added into a 384-hole plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
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TargetHepatocyte growth factor receptor(Human)
Lanova Medicines

US Patent
LigandPNGBDBM477047(US10882853, Compound 24)
Affinity DataIC50: 25.2nMAssay Description:1. Methods(1) 4 μL of prepared kinase buffer solution or 4 μL of kinase solution (100% inhibition control) were added into a 384-hole plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
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TargetVascular endothelial growth factor receptor 2(Human)
Lanova Medicines

US Patent
LigandPNGBDBM477045(US10882853, Compound 5)
Affinity DataIC50: 39.9nMAssay Description:1. Methods(1) 4 μL of prepared kinase buffer solution or 4 μL of kinase solution (100% inhibition control) were added into a 384-hole plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
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TargetVascular endothelial growth factor receptor 2(Human)
Lanova Medicines

US Patent
LigandPNGBDBM477044(US10882853, Compound 10)
Affinity DataIC50: 64.2nMAssay Description:1. Methods(1) 4 μL of prepared kinase buffer solution or 4 μL of kinase solution (100% inhibition control) were added into a 384-hole plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
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TargetHepatocyte growth factor receptor(Human)
Lanova Medicines

US Patent
LigandPNGBDBM477043(US10882853, Compound For-Methyl)
Affinity DataIC50: 163nMAssay Description:1. Methods(1) 4 μL of prepared kinase buffer solution or 4 μL of kinase solution (100% inhibition control) were added into a 384-hole plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2021
Entry Details
Go to US Patent