Compile Data Set for Download or QSAR
Report error Found 693 Enz. Inhib. hit(s) with all data for entry = 9478
TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469350(cis-5-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  0.300nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469376(cis-1-(Cyclobutyl-methyl)-8-dimethylamino-8-phenyl...)
Affinity DataKi:  0.400nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469352(cis-5-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  0.400nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469357(cis-2-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  0.600nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469437(cis-5-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  0.600nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469382(cis-4-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  0.600nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469435(cis-1-(Cyclobutyl-methyl)-8-dimethylamino-3-(2-met...)
Affinity DataKi:  0.600nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469419(cis-5-[1-[(1-Cyano-cyclobutyl)-methyl]-8-dimethyla...)
Affinity DataKi:  0.700nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469354(cis-5-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  0.700nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469365(cis-2-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  0.800nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469398(cis-5-[1-[(1-Cyano-cyclobutyl)-methyl]-8-dimethyla...)
Affinity DataKi:  0.900nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469458(cis-8-Dimethylamino-1-[(1-hydroxy-cyclobutyl)-meth...)
Affinity DataKi:  1nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469378(cis-5-[8-Dimethylamino-1-(2-methyl-propy1)-2-oxo-8...)
Affinity DataKi:  1nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469405(cis-4-[1-(Cyclobuty1-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  1nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469432(cis-1-(Cyclobutyl-methyl)-8-dimethylamino-8-phenyl...)
Affinity DataKi:  1nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469461(cis-1-(Cyclobutyl-methyl)-8-dimethylamino-3-[4-met...)
Affinity DataKi:  1nMAssay Description:The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl (pH 7.4)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469395(cis-1-(Cyclobutyl-methyl)-8-methylamino-8-phenyl-3...)
Affinity DataKi:  1nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469460(cis-1-[(1-Hydroxy-cyclobutyl)-methyl]-8-methylamin...)
Affinity DataKi:  1nMAssay Description:The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl (pH 7.4)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469458(cis-8-Dimethylamino-1-[(1-hydroxy-cyclobutyl)-meth...)
Affinity DataKi:  1nMAssay Description:The hMOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl (pH 7.4)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469708(US10807988, Example SC_3344 | cis-8-Dimethylamino-...)
Affinity DataKi:  1nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469764(US10807988, Example SC_3401 | cis-1-(Cyclobutyl-me...)
Affinity DataKi:  1nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469459(cis-1-[(1-Hydroxy-cyclobutyl1)-methyl]-8-methylami...)
Affinity DataKi:  1nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469358(cis-2-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  1.10nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469355(cis-5-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  1.10nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469445(cis-1-(Cyclobutyl-methyl)-3-(2,4-dimethoxy-phenyl)...)
Affinity DataKi:  1.10nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469452(cis-2-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  1.10nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469351(cis-5-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  1.30nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469449(cis-2-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  1.30nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469364(cis-5-[8-Dimethylamino-1-[(1-hydroxy-cyclobutyl)-m...)
Affinity DataKi:  1.40nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469392(cis-5-[8-Dimethylamino-1-](1-methyl-cyclobutyl)-me...)
Affinity DataKi:  1.40nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469433(cis-5-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  1.60nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469439(cis-4-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  1.60nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469438(cis-1-(Cyclobutyl-methyl)-8-dimethylamino-3-(5-flu...)
Affinity DataKi:  1.60nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469444(cis-1-(Cyclobutyl-methyl)-8-dimethylamino-8-phenyl...)
Affinity DataKi:  1.60nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469374(cis-4-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  1.80nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469383(cis-4-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  1.80nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469443(cis-1-(Cyclobutyl-methyl)-8-dimethylamino-3-[2-met...)
Affinity DataKi:  1.80nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469370(cis-4-[1-(Cyclobutyl-methyl)-8-dimethylamino-2-oxo...)
Affinity DataKi:  2nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469673(US10807988, Example SC_3308 | cis-8-Dimethylamino-...)
Affinity DataKi:  2nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469729(US10807988, Example SC_3365 | cis-8-Dimethylamino-...)
Affinity DataKi:  2nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469456(cis-8-Dimethylamino-1-[(1-hydroxy-cyclobutyl)-meth...)
Affinity DataKi:  2nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469469(cis-1-(Cyclopropyl-methyl)-8-dimethylamino-3-(2-fl...)
Affinity DataKi:  2nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469752(US10807988, Example SC_3389 | cis-3-[6-(Azetidin-1...)
Affinity DataKi:  2nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469695(US10807988, Example SC_3331 | cis-8-Dimethylamino-...)
Affinity DataKi:  2nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469465(cis-1-(Cyclopropyl-methyl)-8-dimethylamino-3-(4-me...)
Affinity DataKi:  2nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469718(US10807988, Example SC_3354 | cis-4-[5-(8-Dimethyl...)
Affinity DataKi:  2nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469750(US10807988, Example SC_3387 | cis-8-Dimethylamino-...)
Affinity DataKi:  2nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469460(cis-1-[(1-Hydroxy-cyclobutyl)-methyl]-8-methylamin...)
Affinity DataKi:  2nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469577(cis-3-(1,3-Benzodioxol-4-yl)-8-dimethylamino-8-phe...)
Affinity DataKi:  2nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetNociceptin receptor(Human)
GrüNenthal

US Patent
LigandPNGBDBM469422(cis-4-[1-(Cyclobutyl-methyl)-8-methylamino-2-oxo-8...)
Affinity DataKi:  2.20nMAssay Description:The hNOP receptor binding assay was performed as homogeneous SPA-assay (scintillation proximity assay) using the assay buffer 50 mM TRIS-HCl. 10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

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