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Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 9471
TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412136(US10392402, Compound A | US10738007, Compound A | ...)
Affinity DataIC50: 2.80nMMore data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412136(US10392402, Compound A | US10738007, Compound A | ...)
Affinity DataIC50: 3.30nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM468965(US10807966, Compound 58)
Affinity DataIC50: 4.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM468967(US10807966, Compound 61)
Affinity DataIC50: 7.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412135(US10392402, Compound ID 52 | US10807966, Compound ...)
Affinity DataIC50: 8.70nMMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM468969(US10807966, Compound 66)
Affinity DataIC50: 9.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM468970(US10807966, Compound 67)
Affinity DataIC50: 10.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412127(US10392402, Compound ID 5 | US10807966, Compound 2...)
Affinity DataIC50: 16.1nMMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412132(US10392402, Compound ID 40 | US10807966, Compound ...)
Affinity DataIC50: 17nMMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM468962(US10807966, Compound 39)
Affinity DataIC50: 17.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM468966(US10807966, Compound 59)
Affinity DataIC50: 20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412130(US10392402, Compound ID 11 | US10807966, Compound ...)
Affinity DataIC50: 22.1nMMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412128(US10392402, Compound ID 7 | US10807966, Compound 7)
Affinity DataIC50: 22.9nMMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM468956(US10807966, Compound 1)
Affinity DataIC50: 27.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412127(US10392402, Compound ID 5 | US10807966, Compound 2...)
Affinity DataIC50: 28.7nMMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM468968(US10807966, Compound 64)
Affinity DataIC50: 29.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412135(US10392402, Compound ID 52 | US10807966, Compound ...)
Affinity DataIC50: 34nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412129(US10392402, Compound ID 9 | US10807966, Compound 9)
Affinity DataIC50: 39.1nMMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412130(US10392402, Compound ID 11 | US10807966, Compound ...)
Affinity DataIC50: 63.6nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM468962(US10807966, Compound 39)
Affinity DataIC50: 65.1nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412127(US10392402, Compound ID 5 | US10807966, Compound 2...)
Affinity DataIC50: 73nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412128(US10392402, Compound ID 7 | US10807966, Compound 7)
Affinity DataIC50: 102nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412127(US10392402, Compound ID 5 | US10807966, Compound 2...)
Affinity DataIC50: 130nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412132(US10392402, Compound ID 40 | US10807966, Compound ...)
Affinity DataIC50: 164nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM468956(US10807966, Compound 1)
Affinity DataIC50: 207nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Translational Drug Development

US Patent
LigandPNGBDBM412129(US10392402, Compound ID 9 | US10807966, Compound 9)
Affinity DataIC50: 237nMAssay Description:The following assay protocol is for measuring the phosphorylation of a peptide substrate (FAM-KKLRRTLSVA-OH wherein FAM is carboxyfluorescein). The p...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Translational Drug Development

US Patent
LigandPNGBDBM468971(US10807966, Compound 68)
Affinity DataIC50: 509nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent