Compile Data Set for Download or QSAR
Report error Found 138 Enz. Inhib. hit(s) with all data for entry = 9454
TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM467005(4-(8-(4-methylphenyl)-5-{[(3R)-1-methylpiperidin-3...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388878(US9944647, Example 3 | 4-(8-(6-methoxypyridin-3-yl...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
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US Patent
LigandPNGBDBM388879(US9944647, Example 4 | 4-(8-[6-(dimethylamino)pyri...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388880(US9944647, Example 5 | 4-[5-{[(3R)-1-methylpiperid...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388882(US9944647, Example 7 | 4-(8-(3-methyl-2-oxo-2,3-di...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
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US Patent
LigandPNGBDBM388883(US9944647, Example 8 | 4-(8-(1-methyl-1H-indazol-5...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
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US Patent
LigandPNGBDBM388884(US9944647, Example 9 | 4-(8-{4-[(4-methylpiperazin...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388885(US9944647, Example 10 | 4-(8-{4-[2-(4-methylpipera...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
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US Patent
LigandPNGBDBM388888(US9944647, Example 13 | (3S)-1-[4-(7-(4-cyanopheny...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388889(US9944647, Example 14 | 4-(8-(4-methyl-3,4-dihydro...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388892(US9944647, Example 17 | 4-(8-(1-methyl-1H-benzimid...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388894(US9944647, Example 19 | 4-[5-{[(3R)-1-methylpiperi...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388895(US9944647, Example 20 | 5-(7-(4-cyanophenyl)-5-{[(...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
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US Patent
LigandPNGBDBM388899(US9944647, Example 24 | 4-(8-(4-methyl-3,4-dihydro...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388906(US9944647, Example 27 | 4-(8-(1-methyl-1H-indazol-...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388907(US9944647, Example 28 | 4-[5-{[(3R)-1-methylpiperi...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388908(US9944647, Example 29 | 4-[5-{[(3R)-1-ethylpiperid...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388909(US9944647, Example 30 | 4-(8-[3-fluoro-4-(hydroxym...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388910(US9944647, Example 31 | 4-(8-[3-fluoro-4-(hydroxym...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388911(US9944647, Example 32 | 4-(8-[3,5-difluoro-4-(hydr...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388912(US9944647, Example 33 | 4-[5-{[(3R)-1-(2-cyanoethy...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388913(US9944647, Example 34 | 4-[5-{[(3R)-1-(2-hydroxyet...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388914(US9944647, Example 35 | 4-(8-[4-(hydroxymethyl)-3-...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388915(US9944647, Example 36 | 4-(8-[4-(hydroxymethyl)phe...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388916(US9944647, Example 37 | 4-[5-[4-(dimethylamino)pip...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388917(US9944647, Example 38 | 4-[5-[(3R)-3-(dimethylamin...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388918(US9944647, Example 39 | 4-[5-(7-methyl-2,7-diazasp...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388920(US9944647, Example 40 | methyl[4-(7-(4-cyanophenyl...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388921(US9944647, Example 41 | 4-[5-{[(3R)-1-(2-methoxyet...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388922(US9944647, Example 42 | 4-(8-(3-amino-1-methyl-1H-...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388923(US9944647, Example 43 | 4-(8-(3-methyl-2-oxo-3,4-d...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388925(US9944647, Example 45 | 4-(8-(5-fluoro-3-methyl-2-...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388926(US9944647, Example 46 | 4-[5-[4-(dimethylamino)pip...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388927(US9944647, Example 47 | 4-[5-[4-(dimethylamino)pip...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388930(US9944647, Example 49 | 4-[5-[4-(dimethylamino)pip...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388932(US9944647, Example 51 | 4-[5-[4-(dimethylamino)pip...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388933(US9944647, Example 52 | 4-{8-[2-(difluoromethyl)-1...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388934(US9944647, Example 53 | 4-[5-[4-(dimethylamino)pip...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388935(US9944647, Example 54 | 4-[5-[4-(dimethylamino)pip...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388936(US9944647, Example 55 | 4-[5-{1[(3R)-1-ethylpiperi...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388937(US9944647, Example 56 | 4-[5-{[(3R)-1-(2-hydroxyet...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388938(US9944647, Example 57 | 4-(8-(5-fluoro-6-methoxypy...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388939(US9944647, Example 58 | 4-[5-[4-(dimethylamino)pip...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388940(US9944647, Example 59 | 4-(8-(4-fluoro-3-methyl-2-...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388941(US9944647, Example 60 | 4-[5-[4-(dimethylamino)pip...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388944(US9944647, Example 62 | 4-[5-[4-(dimethylamino)pip...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388946(US9944647, Example 63 | 4-[5-[4-(dimethylamino)pip...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
Go to US Patent

TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388947(US9944647, Example 64 | 4-(8-[2-(difluoromethyl)-1...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
Go to US Patent

TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388948(US9944647, Example 65 | 4-(8-(1,2-dimethyl-1H-benz...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
Go to US Patent

TargetLysine-specific histone demethylase 1A(Human)
Incyte

US Patent
LigandPNGBDBM388953(US9944647, Example 68 | 4-[5-[4-(dimethylamino)pip...)
Affinity DataIC50: 50nMAssay Description:LANCE LSD1/KDM1A demethylase assay 10 μL of 1 nM LSD-1 enzyme (ENZO BML-SE544-0050) in the assay buffer (50 mM Tris, pH 7.5, 0.01% Tween-20, 25 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
Go to US Patent

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