Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 9413
TargetProstacyclin receptor(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM464509(US10793529, Compound 69 | 2-(((1s,4s)-4-((6-(4- me...)
Affinity DataEC50:  8nMAssay Description:The HTRF assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total volume...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
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TargetProstacyclin receptor(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM464510(US10793529, Compound 31 | 2-(((1s,4s,)-4-((4-(3-ch...)
Affinity DataEC50:  31nMAssay Description:The HTRF assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total volume...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetProstacyclin receptor(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM464511(US10793529, Compound 43 | 2-(((1s,4s)-4-((3-oxo-5,...)
Affinity DataEC50:  36nMAssay Description:The HTRF assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total volume...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent

TargetProstacyclin receptor(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM464512(US10793529, Compound 67 | 2-(((1s,4s)-4-((5-(3- ch...)
Affinity DataEC50:  73nMAssay Description:The HTRF assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total volume...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2021
Entry Details
Go to US Patent