Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 9263
TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM437978(US10618886, Compound I | US10730853, Compound I | ...)
Affinity DataIC50: 1.73nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM437978(US10618886, Compound I | US10730853, Compound I | ...)
Affinity DataIC50: 3.05nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438108(US10618886, Compound II | US10730853, Compound XII...)
Affinity DataIC50: 3.18nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438114(US10618886, Compound VII | US10730853, Compound VI...)
Affinity DataIC50: 3.44nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438108(US10618886, Compound II | US10730853, Compound XII...)
Affinity DataIC50: 3.63nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438112(US10618886, Compound VI | US10730853, Compound IX ...)
Affinity DataIC50: 3.83nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438110(US10618886, Compound IV | US10730853, Compound IV ...)
Affinity DataIC50: 3.87nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438115(US10618886, Compound VIII | US10730853, Compound V...)
Affinity DataIC50: 4.81nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438108(US10618886, Compound II | US10730853, Compound XII...)
Affinity DataIC50: 4.97nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM453705(US10730853, Compound VI | US11420955, Compound VI)
Affinity DataIC50: 5.36nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM453705(US10730853, Compound VI | US11420955, Compound VI)
Affinity DataIC50: 5.5nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438120(US10618886, Compound XIII | US10730853, Compound X...)
Affinity DataIC50: 5.63nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438115(US10618886, Compound VIII | US10730853, Compound V...)
Affinity DataIC50: 6.11nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438112(US10618886, Compound VI | US10730853, Compound IX ...)
Affinity DataIC50: 7.70nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438110(US10618886, Compound IV | US10730853, Compound IV ...)
Affinity DataIC50: 8.15nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438117(US10618886, Compound X | US10730853, Compound X | ...)
Affinity DataIC50: 9.10nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438114(US10618886, Compound VII | US10730853, Compound VI...)
Affinity DataIC50: 10.5nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438120(US10618886, Compound XIII | US10730853, Compound X...)
Affinity DataIC50: 10.9nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438108(US10618886, Compound II | US10730853, Compound XII...)
Affinity DataIC50: 17.6nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438111(US10618886, Compound IX | US10618886, Compound V |...)
Affinity DataIC50: 20nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438109(US10618886, Compound III | US10730853, Compound II...)
Affinity DataIC50: 21.2nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438111(US10618886, Compound IX | US10618886, Compound V |...)
Affinity DataIC50: 36.5nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438109(US10618886, Compound III | US10730853, Compound II...)
Affinity DataIC50: 39.6nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438125(US10618886, Compound XX | US10730853, Compound XX ...)
Affinity DataIC50: 50.5nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438117(US10618886, Compound X | US10730853, Compound X | ...)
Affinity DataIC50: 52.5nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM453716(US10730853, Compound XIV | US11420955, Compound XI...)
Affinity DataIC50: 55.7nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM453716(US10730853, Compound XIV | US11420955, Compound XI...)
Affinity DataIC50: 61.9nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM453717(US10730853, Compound XVI | US11420955, Compound XV...)
Affinity DataIC50: 116nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM453717(US10730853, Compound XVI | US11420955, Compound XV...)
Affinity DataIC50: 175nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438127(US10618886, Compound XXII | US10730853, Compound X...)
Affinity DataIC50: 229nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438127(US10618886, Compound XXII | US10730853, Compound X...)
Affinity DataIC50: 242nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438126(US10618886, Compound XXI | US10730853, Compound XX...)
Affinity DataIC50: 286nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438125(US10618886, Compound XX | US10730853, Compound XX ...)
Affinity DataIC50: 814nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438124(US10618886, Compound XIX | US10730853, Compound XI...)
Affinity DataIC50: 1.00E+3nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438124(US10618886, Compound XIX | US10730853, Compound XI...)
Affinity DataIC50: 1.00E+3nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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TargetHistamine H3 receptor(Human)
Xw Laboratories

US Patent
LigandPNGBDBM438126(US10618886, Compound XXI | US10730853, Compound XX...)
Affinity DataIC50: 1.00E+3nMAssay Description:Materials: GTPγS, [35S] (PerkinElmer, Cat # NEG030H001MC), DMSO (Amresco, Cat #0231), MicroScint™-20 (PerkinElmer, Cat #6013621), CelLytic&...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
Go to US Patent