Compile Data Set for Download or QSAR
Report error Found 423 Enz. Inhib. hit(s) with all data for entry = 11385
LigandPNGBDBM611197((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[3-[5...)
Affinity DataIC50: 0.380nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611196((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[3-[6...)
Affinity DataIC50: 0.410nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611264((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[3-[4...)
Affinity DataIC50: 0.480nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611235((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[2-[4...)
Affinity DataIC50: 0.610nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611236((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[2-[4...)
Affinity DataIC50: 0.610nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611331((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[6-[6...)
Affinity DataIC50: 0.660nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611205((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[2-[4...)
Affinity DataIC50: 0.760nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611240((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[2-[6...)
Affinity DataIC50: 0.830nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611265((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[3-[4...)
Affinity DataIC50: 0.830nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611198((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[6-[4...)
Affinity DataIC50: 0.840nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611330((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[4-[5...)
Affinity DataIC50: 0.880nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611245((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[2-[2...)
Affinity DataIC50: 0.970nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611095((2S)-N-[[3-[(4-cyanophenyl) methoxy]phenyl]methyl]...)
Affinity DataIC50: 1nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611192((2S)-1-(benzofuran-2-ylsulfonyl)- N-[[3-[5-(triflu...)
Affinity DataIC50: 1.20nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611193((2S)-1-(benzofuran-2-ylsulfonyl)- N-[[6-[4-(triflu...)
Affinity DataIC50: 1.20nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611366((1S,3S,5S)-4-(5- fluorobenzofuran-2-yl)sulfonyl- N...)
Affinity DataIC50: 1.20nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611154((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[3-[[...)
Affinity DataIC50: 1.30nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611286((2S)-1-(benzofuran-2- ylsulfonyl)-N-[[4-[5- (trifl...)
Affinity DataIC50: 1.30nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611332((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[4-[5...)
Affinity DataIC50: 1.30nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611133((2S)-1-(5-fluorobenzofuran- 2-yl)sulfonyl-N-[[3-[[...)
Affinity DataIC50: 1.40nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611396((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[6-[2...)
Affinity DataIC50: 1.40nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611149((2S)-N-[[3-[(4- cyanophenyl)methoxy]- 5-fluoro- ph...)
Affinity DataIC50: 1.5nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611256((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[4-[6...)
Affinity DataIC50: 1.5nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611147((2S)-N-[(3-benzyloxy-5- fluoro-phenyl)methyl]- 1-(...)
Affinity DataIC50: 1.60nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611156((2S)-N-[(3-benzyloxyphenyl) methyl]-1-(5-fluoroben...)
Affinity DataIC50: 1.60nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611191((2S)-1-(benzofuran-2-ylsulfonyl)- N-[[3-[6-(triflu...)
Affinity DataIC50: 1.60nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611207((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[3-[6...)
Affinity DataIC50: 1.60nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611380((2S)-1-furo[3,2-c]pyridin-2- ylsulfonyl-N-[[4-hydr...)
Affinity DataIC50: 1.60nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611157((2S)-1-(benzofuran-2- ylsulfonyl)-N-[[3-[[4- (trif...)
Affinity DataIC50: 1.70nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611413((2S)-1-(benzofuran-2-ylsulfonyl)-N-[[4- fluoro-3-[...)
Affinity DataIC50: 1.70nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611258((2S)-1-(benzofuran-2- ylsulfonyl)-N-[[4-[6- (trifl...)
Affinity DataIC50: 1.90nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611365((1R,3S,5R)-4-(5- fluorobenzofuran-2-yl)sulfonyl- N...)
Affinity DataIC50: 1.90nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611237((2S)-N-[[2-[4- (difluoromethoxy)phenyl]-4- pyridyl...)
Affinity DataIC50: 2nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611263((2S)-N-[[3-(4- chlorophenyl)phenyl]methyl]-1- (5-f...)
Affinity DataIC50: 2.10nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611322((2S)-1-(benzofuran-2- ylsulfonyl)-N-[[5-hydroxy-4-...)
Affinity DataIC50: 2.10nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611199((2S)-1-(4-fluorobenzofuran-2- yl)sulfonyl-N-[[3-[6...)
Affinity DataIC50: 2.20nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611247((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[5-[6...)
Affinity DataIC50: 2.20nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611255((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[4-[4...)
Affinity DataIC50: 2.20nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611300(Synthesis of (2S)-1-(benzofuran-2-ylsulfonyl)-N-[[...)
Affinity DataIC50: 2.20nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611369((1S,2S,4R)-3-(5- fluorobenzofuran-2-yl)sulfonyl- N...)
Affinity DataIC50: 2.30nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611222((2S)-1-(benzofuran-2- ylsulfonyl)-N-[[2-[4- (trifl...)
Affinity DataIC50: 2.40nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611329((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[4-[4...)
Affinity DataIC50: 2.40nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611302((2S)-1-(benzofuran-2- ylsulfonyl)-N-[[3-[2- (trifl...)
Affinity DataIC50: 2.5nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611395((2S)-1-(benzofuran-2-ylsulfonyl)-N- [[6-[2-hydroxy...)
Affinity DataIC50: 2.5nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611416(Synthesis of (2S)-1-(benzofuran-2-ylsulfonyl)-N-[[...)
Affinity DataIC50: 2.5nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611505((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[3-[5...)
Affinity DataIC50: 2.5nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611230((2S)-1-(benzofuran-2- ylsulfonyl)-N-[[2-[2-hydroxy...)
Affinity DataIC50: 2.60nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611166((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[3-[4...)
Affinity DataIC50: 2.70nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611494((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[6-[6...)
Affinity DataIC50: 2.70nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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LigandPNGBDBM611512((2S)-1-(5-fluorobenzofuran-2- yl)sulfonyl-N-[[6-[4...)
Affinity DataIC50: 2.70nMAssay Description:The test substance was dissolved in dimethyl sulfoxide and serially diluted with an assay buffer containing 0.1% bovine serum albumin (1×HBSS, 20 mM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2023
Entry Details
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