Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 8969
LigandPNGBDBM433319(US10561656, Example 2 | 3-(ethylthio)-2-(4-(6-fluo...)
Affinity DataIC50: 1nMAssay Description:Assay: The following phosphodiesterase enzymes may be used: 3′,5′-cyclic-nucleotide-specific bovine brain phosphodiesterase (Sigma, St. L...More data for this Ligand-Target Pair
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Date in BDB:
11/22/2020
Entry Details
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LigandPNGBDBM433321(US10561656, Example 3-A | (6aR,9aS)-5,6a,7,8,9,9a-...)
Affinity DataIC50: 1.5nMAssay Description:Assay: The following phosphodiesterase enzymes may be used: 3′,5′-cyclic-nucleotide-specific bovine brain phosphodiesterase (Sigma, St. L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
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LigandPNGBDBM433318(US10561656, Example 1 | 3-(ethylthio)-2-(4-(5-fluo...)
Affinity DataIC50: 2.70nMAssay Description:Assay: The following phosphodiesterase enzymes may be used: 3′,5′-cyclic-nucleotide-specific bovine brain phosphodiesterase (Sigma, St. L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
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LigandPNGBDBM433320(US10561656, Example 3 | 2-(4-(6-fluoropyridin-2-yl...)
Affinity DataIC50: 5nMAssay Description:Assay: The following phosphodiesterase enzymes may be used: 3′,5′-cyclic-nucleotide-specific bovine brain phosphodiesterase (Sigma, St. L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
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LigandPNGBDBM433322(US10561656, Example 3-B | (6aR,9aS)-5,6a,7,8,9,9a-...)
Affinity DataIC50: 6nMAssay Description:Assay: The following phosphodiesterase enzymes may be used: 3′,5′-cyclic-nucleotide-specific bovine brain phosphodiesterase (Sigma, St. L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
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LigandPNGBDBM433320(US10561656, Example 3 | 2-(4-(6-fluoropyridin-2-yl...)
Affinity DataIC50: 3.00E+3nMAssay Description:Assay: The following phosphodiesterase enzymes may be used: 3′,5′-cyclic-nucleotide-specific bovine brain phosphodiesterase (Sigma, St. L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
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LigandPNGBDBM433319(US10561656, Example 2 | 3-(ethylthio)-2-(4-(6-fluo...)
Affinity DataIC50: 4.00E+3nMAssay Description:Assay: The following phosphodiesterase enzymes may be used: 3′,5′-cyclic-nucleotide-specific bovine brain phosphodiesterase (Sigma, St. L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
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LigandPNGBDBM433318(US10561656, Example 1 | 3-(ethylthio)-2-(4-(5-fluo...)
Affinity DataIC50: 1.10E+4nMAssay Description:Assay: The following phosphodiesterase enzymes may be used: 3′,5′-cyclic-nucleotide-specific bovine brain phosphodiesterase (Sigma, St. L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
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LigandPNGBDBM433321(US10561656, Example 3-A | (6aR,9aS)-5,6a,7,8,9,9a-...)
Affinity DataIC50: 2.70E+4nMAssay Description:Assay: The following phosphodiesterase enzymes may be used: 3′,5′-cyclic-nucleotide-specific bovine brain phosphodiesterase (Sigma, St. L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
Go to US Patent