Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 8932
LigandPNGBDBM430025(US10538523, Example 1 | 4-(4′-Ethanesulfonyl...)
Affinity DataKi: <0.600nMAssay Description:The affinity of the test compounds was determined by radioligand competition binding assay, using the known compound [3H]Ro-15-1788 (Flumazenil) (Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2020
Entry Details
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LigandPNGBDBM430027(US10538523, Example 3 | 5-[5-(1-Ethyl-1H-pyrazolo[...)
Affinity DataKi:  11.8nMAssay Description:The affinity of the test compounds was determined by radioligand competition binding assay, using the known compound [3H]Ro-15-1788 (Flumazenil) (Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2020
Entry Details
Go to US Patent

LigandPNGBDBM430026(US10538523, Example 2 | 4-(4′-Ethanesulfonyl...)
Affinity DataKi:  17.5nMAssay Description:The affinity of the test compounds was determined by radioligand competition binding assay, using the known compound [3H]Ro-15-1788 (Flumazenil) (Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2020
Entry Details
Go to US Patent