Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with all data for entry = 8878
TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM314726(US9611269, Example 39 | US10513522, Example 39 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314690(US9611269, Example 3 | US10513522, Example 27 | US...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314725(US9611269, Example 38 | US10513522, Example 38 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314713(US9611269, Example 26 | US10513522, Example 26 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314712(US9611269, Example 25 | US10513522, Example 25 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314712(US9611269, Example 25 | US10513522, Example 25 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314711(US9611269, Example 24 | US10513522, Example 24 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314711(US9611269, Example 24 | US10513522, Example 24 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314710(US9611269, Example 23 | US10513522, Example 23 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314690(US9611269, Example 3 | US10513522, Example 27 | US...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314709(US9611269, Example 22 | US10513522, Example 22 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314708(US9611269, Example 21 | US10513522, Example 21 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314708(US9611269, Example 21 | US10513522, Example 21 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314707(US9611269, Example 20 | US10513522, Example 20 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314727(US9611269, Example 40 | US10513522, Example 40 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314706(US9611269, Example 19 | US10513522, Example 19 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM246876(US10053465, 15 | US10053465, 17 | 5-{3-(cyanomethy...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314688(US9611269, Example 1 | US10513522, Example 1 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM246877(4-{3-(cyanomethyl)- 3-[4-(7H-pyrrolo[2,3- d]pyrimi...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM246877(4-{3-(cyanomethyl)- 3-[4-(7H-pyrrolo[2,3- d]pyrimi...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314716(US9611269, Example 29 | US10513522, Example 29 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314716(US9611269, Example 29 | US10513522, Example 29 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314717(US9611269, Example 30 | US10513522, Example 30 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314724(US9611269, Example 37 | US10513522, Example 37 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314718(US9611269, Example 31 | US10513522, Example 31 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK2(Human)
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US Patent
LigandPNGBDBM314718(US9611269, Example 31 | US10513522, Example 31 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314719(US9611269, Example 32 | US10513522, Example 32 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314719(US9611269, Example 32 | US10513522, Example 32 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314720(US9611269, Example 33 | US10513522, Example 33 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314724(US9611269, Example 37 | US10513522, Example 37 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM262166(5-{3-(cyanomethyl)- 3-[4-(1H-pyrrolo[2,3- b]pyridi...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314722(US9611269, Example 35 | US10513522, Example 35 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314723(US9611269, Example 36 | US10513522, Example 36 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314693(US9611269, Example 6 | US10513522, Example 6 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314697(US9611269, Example 10 | US10513522, Example 10 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314696(US9611269, Example 9 | US10513522, Example 9 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM314696(US9611269, Example 9 | US10513522, Example 9 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314695(US9611269, Example 8 | US10513522, Example 8 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM314695(US9611269, Example 8 | US10513522, Example 8 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314694(US9611269, Example 7 | US10513522, Example 7 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM314694(US9611269, Example 7 | US10513522, Example 7 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314693(US9611269, Example 6 | US10513522, Example 6 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314704(US9611269, Example 17 | US10513522, Example 17 | U...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314692(US9611269, Example 5 | US10513522, Example 5 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314692(US9611269, Example 5 | US10513522, Example 5 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314691(US9611269, Example 4 | US10513522, Example 4 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314691(US9611269, Example 4 | US10513522, Example 4 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314690(US9611269, Example 3 | US10513522, Example 27 | US...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM314690(US9611269, Example 3 | US10513522, Example 27 | US...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
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LigandPNGBDBM314689(US9611269, Example 2 | US10513522, Example 2 | US1...)
Affinity DataIC50: 10nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
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