Compile Data Set for Download or QSAR
Report error Found 196 Enz. Inhib. hit(s) with all data for entry = 8646
TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344018(US9777017, Example 10 | US9777017, Example 2 | US9...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344020(US9777017, Example 4 | US9908895, Example 4 | US10...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344021(US9777017, Example 5 | US9908895, Example 5 | US10...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344023(US9777017, Example 7 | US9908895, Example 7 | US10...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344024(US9777017, Example 8 | US9908895, Example 8 | US10...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344018(US9777017, Example 10 | US9777017, Example 2 | US9...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344027(US9777017, Example 11 | US9908895, Example 11 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344028(US9777017, Example 12 | US9908895, Example 12 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344029(US9777017, Example 13 | US9908895, Example 13 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344033(US9777017, Example 17 | US9908895, Example 17 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344034(US9777017, Example 18 | US9908895, Example 18 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM246852(((2R,5S)-5-{2-[(1R)- 1-hydroxyethyl]-1H- imidazo[4...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344039(US9777017, Example 23 | US10370387, Example 23 | U...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344040(US9777017, Example 24 | US9908895, Example 24 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344041(US9777017, Example 25 | US9908895, Example 25 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344042(US9777017, Example 26 | US9908895, Example 26 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344043(US9777017, Example 27 | US9908895, Example 27 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344048(US9777017, Example 32 | US9908895, Example 32 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344049(US9777017, Example 33 | US9908895, Example 33 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344051(US9777017, Example 35 | US9908895, Example 35 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM410241(((1R,2R,4S)-2-Hydroxy-4-{2-[(1R)-1-hydroxyethyl]-1...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM410242(US10370387, Example 37-2 | US10370387, Example 36-...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM410242(US10370387, Example 37-2 | US10370387, Example 36-...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344054(US9777017, Example 38 | US9908895, Example 38 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK2 [828-1132](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344054(US9777017, Example 38 | US9908895, Example 38 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344055(US9777017, Example 39 | US9908895, Example 39 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM375666(US9908895, Example 40 | US9908895, Example 41 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM410249([(1R,2S,4S)-4-(2-Methyl-1H-imidazo[4,5-d]thieno[3,...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344058(US9777017, Example 42 | US9908895, Example 42 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344059(US9777017, Example 43 | US9908895, Example 43 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344061(US9777017, Example 45 | US9908895, Example 45 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM410255([4-(8-Methylpyrazolo[1,5-c]thieno[2,3-e]pyrimidin-...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344063(US9777017, Example 47 | US9908895, Example 47 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344064(US9777017, Example 48 | US9908895, Example 48 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK2 [828-1132](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344064(US9777017, Example 48 | US9908895, Example 48 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344073(US9777017, Example 57 | US9908895, Example 57 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344074(US9777017, Example 58 | US9908895, Example 58 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344080(US9777017, Example 64 | US9908895, Example 64 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344084(US9777017, Example 68 | US10370387, Example 68 | U...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344087(US9777017, Example 71 | US9908895, Example 71 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344088(US9777017, Example 72 | US9908895, Example 72 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344089(US9777017, Example 73 | US9908895, Example 73 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344091(US9777017, Example 75 | US9908895, Example 75 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344092(US9777017, Example 76 | US9908895, Example 76 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344093(US9777017, Example 77 | US9908895, Example 77 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK2 [828-1132](Human)
Incyte Holdings

US Patent
LigandPNGBDBM344093(US9777017, Example 77 | US9908895, Example 77 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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LigandPNGBDBM410287(Methyl [(trans-4-{2-[(1R)-1-hydroxyethyl]-1H-imida...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344095(US9777017, Example 79 | US9908895, Example 79 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344096(US9777017, Example 80 | US9908895, Example 80 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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TargetTyrosine-protein kinase JAK1 [837-1142](Human)
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US Patent
LigandPNGBDBM344097(US9777017, Example 81 | US9908895, Example 81 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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