Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 8637
LigandPNGBDBM409965(4-(cycloheptyl- oxy)-2-oxo-1,2- dihydro- quinoline...)
Affinity DataKi:  29nMAssay Description:Human PDE9 (PDE9A2, GenBank Accession No. NM_001001567), full length with N-terminal GST tag, was purchased from BPS Bioscience. The fluorescence pol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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LigandPNGBDBM409964(US10370337, Example 1-7)
Affinity DataKi:  50.3nMAssay Description:Human PDE9 (PDE9A2, GenBank Accession No. NM_001001567), full length with N-terminal GST tag, was purchased from BPS Bioscience. The fluorescence pol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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LigandPNGBDBM409968(4-((3-allyl- oxetan-3-yl) methoxy)-2- oxo-1,2- dih...)
Affinity DataKi:  87.8nMAssay Description:Human PDE9 (PDE9A2, GenBank Accession No. NM_001001567), full length with N-terminal GST tag, was purchased from BPS Bioscience. The fluorescence pol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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LigandPNGBDBM409966(2-oxo-4- tetrahydropyran- 4-yloxy-1H- quinoline- 3...)
Affinity DataKi:  135nMAssay Description:Human PDE9 (PDE9A2, GenBank Accession No. NM_001001567), full length with N-terminal GST tag, was purchased from BPS Bioscience. The fluorescence pol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
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LigandPNGBDBM409967(2-oxo-4-(2- hydroxymethyl- 2-methyl-1- butyloxy)- ...)
Affinity DataKi:  182nMAssay Description:Human PDE9 (PDE9A2, GenBank Accession No. NM_001001567), full length with N-terminal GST tag, was purchased from BPS Bioscience. The fluorescence pol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent