Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 8605
TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406684(1-(4-(7-(4-(pyridin-2-oxy)phenyl)-1H-pyrazazo[3,4-...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406695(US10336755, Example 22b)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406694(US10336755, Example 22a)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406693(1-(2-(7-(4-phenoxyphenyl)-1H-pyrazolo[3,4-c]pyridi...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406692(1-(3-(7-(4-phenoxyphenyl)-1H-indazol-5-yl)piperidi...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406690(4-(5-(1-acryloylpyrrolidin-3-yl)-1H-pyrazolo[3,4-c...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406687(1-(4-(7-(4-(3-fluorophenoxyl)phenyl)-1H-pyrazolo[3...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406686(1-(4-(7-(2-fluoro-4-phenoxyphenyl)-1H-pyrazolo[3,4...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406685(1-(4-(7-(4-(pyridin-2-oxy)phenyl)-1H-pyrazolo[3,4-...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406683(1-(3-((7-(4-phenoxyphenyl)-1H-pyrazolo[3,4-c]pyrid...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406682(N-(1-(7-(4-phenoxyphenyl)-1H-pyrazolo[3,4-c]pyridi...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406681(1-(4-(7-(4-phenoxyphenyl)-1H-pyrazolo[3,4-c]pyridi...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406680(N-(3-(7-(4-phenoxyphenyl)-1H-pyrazolo[3,4-c]pyridi...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406675(1-(4-(7-(4-phenoxyphenyl)-1H-pyrazolo[3,4-c]pyridi...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406674(1-(3-(7-(4-phenoxyphenyl)-1H-pyrazolo[3,4-c]pyridi...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406673(7-(4-phenoxyphenyl)-5-(1-(ethenylsulfonyl)piperidi...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406672((E)-4-(dimethylamino)-1-(3-(7-(4-phenoxyphenyl)-1H...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406671(1-(3-(7-(4-phenoxyphenyl)-1H-pyrazolo[3,4-c]pyridi...)
Affinity DataIC50: 100nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406669(1-(3-(7-(4-(morpholinomethyl)phenyl)-1H-pyrazolo[3...)
Affinity DataIC50: 300nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406689(1-(3-(7-(4-phenoxyphenyl)-1H-pyrazolo[3,4-c]pyridi...)
Affinity DataIC50: 300nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406691(4-(5-(1-(but-2-ynoyl)pyrrolidin-3-yl)-1H-pyrazolo[...)
Affinity DataIC50: 300nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406670(1-(3-(7-(4-(oxetan-3-oxy)phenyl)-1H-pyrazolo[3,4-c...)
Affinity DataIC50: 300nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK(Human)
Beijing Innocare Pharma Tech

US Patent
LigandPNGBDBM406688(1-(4-(7-(4-(pyrrolidin-1-ylmethyl)phenyl)-1H-pyraz...)
Affinity DataIC50: 500nMAssay Description:In vitro activity of BTK is measured by detecting ADP produced in a kinase reaction with an ADP-Glo kinase assay kit from Promega Company. In the kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2020
Entry Details
Go to US Patent