Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 3382
TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266567(US10323016, Example 21 | CHEMBL4090147)
Affinity DataEC50:  35nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
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TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266572(US10323016, Example 15 | CHEMBL4060122)
Affinity DataEC50:  370nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
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TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266557(US10323016, Example 16 | CHEMBL4063932)
Affinity DataEC50:  990nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
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TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266557(US10323016, Example 16 | CHEMBL4063932)
Affinity DataEC50:  90nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
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TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266565(US10323016, Example 17 | CHEMBL4091702)
Affinity DataEC50:  1.10E+3nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
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TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266565(US10323016, Example 17 | CHEMBL4091702)
Affinity DataEC50:  140nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
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TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266558(US10323016, Example 18 | CHEMBL4088938)
Affinity DataEC50:  750nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266558(US10323016, Example 18 | CHEMBL4088938)
Affinity DataEC50:  510nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
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TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266566(US10323016, Example 19 | CHEMBL4068227)
Affinity DataEC50:  47nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
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TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266566(US10323016, Example 19 | CHEMBL4068227)
Affinity DataEC50:  4.80nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266552(US10323016, Example 20 | CHEMBL4094487)
Affinity DataEC50:  15nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
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TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266552(US10323016, Example 20 | CHEMBL4094487)
Affinity DataEC50:  1nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266572(US10323016, Example 15 | CHEMBL4060122)
Affinity DataEC50:  900nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266567(US10323016, Example 21 | CHEMBL4090147)
Affinity DataEC50:  2nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
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TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398283(US10323016, Example 22)
Affinity DataEC50:  580nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398283(US10323016, Example 22)
Affinity DataEC50:  29nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398284(US10323016, Example 23)
Affinity DataEC50:  330nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398284(US10323016, Example 23)
Affinity DataEC50:  26nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398285(US10323016, Example 24)
Affinity DataEC50:  1.20E+3nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398285(US10323016, Example 24)
Affinity DataEC50:  68nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398286(US10323016, Example 25)
Affinity DataEC50:  240nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398286(US10323016, Example 25)
Affinity DataEC50:  10nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398287(US10323016, Example 26)
Affinity DataEC50:  40nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398287(US10323016, Example 26)
Affinity DataEC50:  0.5nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398270(US10323016, Example 7)
Affinity DataEC50:  177nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266536(US10323016, Example 1 | CHEMBL4085664)
Affinity DataEC50:  68nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266574(US10323016, Example 2 | CHEMBL4081298)
Affinity DataEC50:  299nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266574(US10323016, Example 2 | CHEMBL4081298)
Affinity DataEC50:  44nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266537(US10323016, Example 3 | CHEMBL4075688)
Affinity DataEC50:  128nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266537(US10323016, Example 3 | CHEMBL4075688)
Affinity DataEC50:  12nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266538(US10323016, Example 4 | CHEMBL4084668)
Affinity DataEC50:  39nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266538(US10323016, Example 4 | CHEMBL4084668)
Affinity DataEC50:  1nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266556(US10323016, Example 5 | CHEMBL4073081)
Affinity DataEC50:  880nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266556(US10323016, Example 5 | CHEMBL4073081)
Affinity DataEC50:  44nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266560(US10323016, Example 6 | CHEMBL4104359)
Affinity DataEC50:  71nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266560(US10323016, Example 6 | CHEMBL4104359)
Affinity DataEC50:  4nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266536(US10323016, Example 1 | CHEMBL4085664)
Affinity DataEC50:  156nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398270(US10323016, Example 7)
Affinity DataEC50:  7nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398271(US10323016, Example 8)
Affinity DataEC50:  260nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398271(US10323016, Example 8)
Affinity DataEC50:  17nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398272(US10323016, Example 9 | US10323016, Example 22 | U...)
Affinity DataEC50:  160nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398272(US10323016, Example 9 | US10323016, Example 22 | U...)
Affinity DataEC50:  18nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266540(US10323016, Example 12 | CHEMBL4102610)
Affinity DataEC50:  4.30E+3nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266540(US10323016, Example 12 | CHEMBL4102610)
Affinity DataEC50:  180nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266573(US10323016, Example 13 | CHEMBL4104779)
Affinity DataEC50:  250nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266573(US10323016, Example 13 | CHEMBL4104779)
Affinity DataEC50:  5nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Human)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266575(US10323016, Example 14 | CHEMBL4085777)
Affinity DataEC50:  7.70E+3nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM50266575(US10323016, Example 14 | CHEMBL4085777)
Affinity DataEC50:  940nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
Go to US Patent