Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 2229
TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357915(US10214536, Compound 275 | (E)-2-(((Dimethylamino)...)
Affinity DataIC50: 80nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357864(US10214536, Compound 24)
Affinity DataIC50: 110nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357870(US10214536, Compound 38)
Affinity DataIC50: 150nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357869(US10214536, Compound 36)
Affinity DataIC50: 160nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357894(US10214536, Compound 76)
Affinity DataIC50: 170nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357919(US10214536, Compound 286)
Affinity DataIC50: 180nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357921(US10214536, Compound 288)
Affinity DataIC50: 180nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357877(US10214536, Compound 53)
Affinity DataIC50: 190nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357872(US10214536, Compound 42)
Affinity DataIC50: 190nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357866(US10214536, Compound 28)
Affinity DataIC50: 220nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357865(US10214536, Compound 26)
Affinity DataIC50: 240nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357871(US10214536, Compound 40)
Affinity DataIC50: 240nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357896(US10214536, Compound 80)
Affinity DataIC50: 260nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357891(US10214536, Compound 69)
Affinity DataIC50: 320nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357897(US10214536, Compound 81)
Affinity DataIC50: 330nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357860(US10214536, Compound 11)
Affinity DataIC50: 340nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357889(US10214536, Compound 65)
Affinity DataIC50: 370nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357929(US10214536, Compound 296)
Affinity DataIC50: 390nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357931(US10214536, Compound 298)
Affinity DataIC50: 410nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357909(US10214536, Compound 258 | 2-Amino-8-isopropyl-5-o...)
Affinity DataIC50: 410nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357893(US10214536, Compound 74)
Affinity DataIC50: 510nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357906(US10214536, Compound 251b | Ethyl 2-amino-8-bromo-...)
Affinity DataIC50: 520nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357930(US10214536, Compound 297)
Affinity DataIC50: 550nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357861(US10214536, Compound 13)
Affinity DataIC50: 560nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357859(US10214536, Compound 8)
Affinity DataIC50: 560nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357892(US10214536, Compound 71)
Affinity DataIC50: 600nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357886(US10214536, Compound 59 | 2-Amino-7-(4,4-dimethylc...)
Affinity DataIC50: 740nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357895(US10214536, Compound 78)
Affinity DataIC50: 790nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357884(US10214536, Compound 57b)
Affinity DataIC50: 800nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357880(US10214536, Compound 55c)
Affinity DataIC50: 880nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357857(US10214536, Amlexanox | Aphthasol)
Affinity DataIC50: 980nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357901(US10214536, Compound 180)
Affinity DataIC50: 1.07E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357887(US10214536, Compound 61)
Affinity DataIC50: 1.17E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357874(US10214536, Compound 47)
Affinity DataIC50: 1.20E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357905(US10214536, Compound 246 | 2-Amino-7-isobutyl-5-ox...)
Affinity DataIC50: 1.23E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357914(US10214536, Compound 272 | 2-Amino-8-fluoro-7-isop...)
Affinity DataIC50: 1.24E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357927(US10214536, Compound 294)
Affinity DataIC50: 1.39E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357922(US10214536, Compound 289)
Affinity DataIC50: 1.40E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357900(US10214536, Compound 176)
Affinity DataIC50: 1.40E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357888(US10214536, Compound 62 | Ethyl 2-amino-7-(4,4-dim...)
Affinity DataIC50: 1.41E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357890(US10214536, Compound 67)
Affinity DataIC50: 1.45E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357907(US10214536, Compound 253b | (E)-2-Amino-8-(2-cyclo...)
Affinity DataIC50: 1.49E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357858(US10214536, Compound 5)
Affinity DataIC50: 1.51E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357932(US10214536, Compound 299)
Affinity DataIC50: 1.53E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357898(US10214536, Compound 97)
Affinity DataIC50: 1.56E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357904(US10214536, Compound 243b | 2-Amino-7-(2-cyclobuty...)
Affinity DataIC50: 1.67E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357862(US10214536, Compound 15)
Affinity DataIC50: 1.67E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357903(US10214536, Compound 243a | 2-Amino-7-isopentyl-5-...)
Affinity DataIC50: 2.01E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357924(US10214536, Compound 291)
Affinity DataIC50: 2.05E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM357912(US10214536, Compound 266b | Ethyl 2-amino-8-fluoro...)
Affinity DataIC50: 2.16E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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