Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 1986
LigandPNGBDBM350000((S)-(4,6-bis(trifluoromethyl)-1H- benzo[d]imidazol...)
Affinity DataIC50: 312nMAssay Description:NAV1.7 SLOW INACTIVATION BLOCK (nM) (Manual Patchclamp).More data for this Ligand-Target Pair
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Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349999((2R)-2-amino-N-(2-(3,5- bis(trifluoromethyl)phenox...)
Affinity DataIC50: 436nMAssay Description:NAV1.7 SLOW INACTIVATION BLOCK (nM) (Manual Patchclamp).More data for this Ligand-Target Pair
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Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349995((R)-2-amino-N-((S)-1-(3,5- bis(trifluoromethyl)phe...)
Affinity DataIC50: 568nMAssay Description:NAV1.7 SLOW INACTIVATION BLOCK (nM) (Manual Patchclamp).More data for this Ligand-Target Pair
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Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349996((2R)-2-amino-N-(1-(3,5- bis(trifluoromethyl)phenox...)
Affinity DataIC50: 1.66E+3nMAssay Description:NAV1.7 INWARD CURRENT BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
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Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349997(2-amino-N-((S)-1-(3,5- bis(trifluoromethyl)phenoxy...)
Affinity DataIC50: 1.89E+3nMAssay Description:NAV1.7 INWARD CURRENT BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349995((R)-2-amino-N-((S)-1-(3,5- bis(trifluoromethyl)phe...)
Affinity DataIC50: 2.58E+3nMAssay Description:NAV1.7 SLOW INACTIVATION BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349996((2R)-2-amino-N-(1-(3,5- bis(trifluoromethyl)phenox...)
Affinity DataIC50: 2.77E+3nMAssay Description:NAV1.7 SLOW INACTIVATION BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
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Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM350000((S)-(4,6-bis(trifluoromethyl)-1H- benzo[d]imidazol...)
Affinity DataIC50: 2.89E+3nMAssay Description:NAV1.7 SLOW INACTIVATION BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349998((R)-N-(2-(3-fluoro-5- (trifluoromethyl)phenoxy)eth...)
Affinity DataIC50: 3.50E+3nMAssay Description:NAV1.7 SLOW INACTIVATION BLOCK (nM) (Manual Patchclamp).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349997(2-amino-N-((S)-1-(3,5- bis(trifluoromethyl)phenoxy...)
Affinity DataIC50: 4.12E+3nMAssay Description:NAV1.7 SLOW INACTIVATION BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
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Date in BDB:
9/21/2019
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LigandPNGBDBM349999((2R)-2-amino-N-(2-(3,5- bis(trifluoromethyl)phenox...)
Affinity DataIC50: 5.32E+3nMAssay Description:NAV1.7 SLOW INACTIVATION BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
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Date in BDB:
9/21/2019
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LigandPNGBDBM349998((R)-N-(2-(3-fluoro-5- (trifluoromethyl)phenoxy)eth...)
Affinity DataIC50: 8.12E+3nMAssay Description:NAV1.7 SLOW INACTIVATION BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349998((R)-N-(2-(3-fluoro-5- (trifluoromethyl)phenoxy)eth...)
Affinity DataIC50: 9.62E+3nMAssay Description:NAV1.7 INWARD CURRENT BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
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Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349999((2R)-2-amino-N-(2-(3,5- bis(trifluoromethyl)phenox...)
Affinity DataIC50: 1.03E+4nMAssay Description:In some cases, the potency of compounds was measured using either the Patchliner automated patch clamp platform (Nanion) or manual patch clamp techni...More data for this Ligand-Target Pair
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Date in BDB:
9/21/2019
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LigandPNGBDBM349997(2-amino-N-((S)-1-(3,5- bis(trifluoromethyl)phenoxy...)
Affinity DataIC50: 1.15E+4nMAssay Description:In some cases, the potency of compounds was measured using either the Patchliner automated patch clamp platform (Nanion) or manual patch clamp techni...More data for this Ligand-Target Pair
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Date in BDB:
9/21/2019
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LigandPNGBDBM349996((2R)-2-amino-N-(1-(3,5- bis(trifluoromethyl)phenox...)
Affinity DataIC50: 1.27E+4nMAssay Description:In some cases, the potency of compounds was measured using either the Patchliner automated patch clamp platform (Nanion) or manual patch clamp techni...More data for this Ligand-Target Pair
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Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349998((R)-N-(2-(3-fluoro-5- (trifluoromethyl)phenoxy)eth...)
Affinity DataIC50: 1.50E+4nMAssay Description:NAV1.7 INWARD CURRENT BLOCK (nM) (0.25HZ Automated Patchclamp).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349998((R)-N-(2-(3-fluoro-5- (trifluoromethyl)phenoxy)eth...)
Affinity DataIC50: 1.50E+4nMAssay Description:In some cases, the potency of compounds was measured using either the Patchliner automated patch clamp platform (Nanion) or manual patch clamp techni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM350001((R)-2-amino-N-((4,6- bis(trifluoromethyl)-1H- benz...)
Affinity DataIC50: 1.50E+4nMAssay Description:NAV1.7 INWARD CURRENT BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM350001((R)-2-amino-N-((4,6- bis(trifluoromethyl)-1H- benz...)
Affinity DataIC50: 1.50E+4nMAssay Description:In some cases, the potency of compounds was measured using either the Patchliner automated patch clamp platform (Nanion) or manual patch clamp techni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM350001((R)-2-amino-N-((4,6- bis(trifluoromethyl)-1H- benz...)
Affinity DataIC50: 1.50E+4nMAssay Description:NAV1.7 SLOW INACTIVATION BLOCK (nM) (Automated Patchclamp).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349995((R)-2-amino-N-((S)-1-(3,5- bis(trifluoromethyl)phe...)
Affinity DataIC50: 1.55E+4nMAssay Description:In some cases, the potency of compounds was measured using either the Patchliner automated patch clamp platform (Nanion) or manual patch clamp techni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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LigandPNGBDBM349998((R)-N-(2-(3-fluoro-5- (trifluoromethyl)phenoxy)eth...)
Affinity DataIC50: 2.32E+4nMAssay Description:NAV1.7 INWARD CURRENT BLOCK (nM) (7HZ Manual Patchclamp).More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
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