Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 1244
TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313753(US10167282, Compound TBAP-04)
Affinity DataIC50: 8nMAssay Description:Mutant BRAF WM266.4 Cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
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TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313751(US10167282, Compound TBAP-02)
Affinity DataIC50: 12nMAssay Description:Mutant BRAF WM266.4 Cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313750(US10167282, Compound TBAP-01)
Affinity DataIC50: 18nMAssay Description:Mutant BRAF WM266.4 Cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313752(US10167282, Compound TBAP-03)
Affinity DataIC50: 19nMAssay Description:Mutant BRAF WM266.4 Cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313753(US10167282, Compound TBAP-04)
Affinity DataIC50: 47nMAssay Description:V600EBRAF was generated by infection of SF9 insect cells cultured in SF-900 II medium (Invitrogen, Paisley, Scotland) with a baculovirus containing f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313750(US10167282, Compound TBAP-01)
Affinity DataIC50: 62nMAssay Description:V600EBRAF was generated by infection of SF9 insect cells cultured in SF-900 II medium (Invitrogen, Paisley, Scotland) with a baculovirus containing f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313751(US10167282, Compound TBAP-02)
Affinity DataIC50: 99nMAssay Description:V600EBRAF was generated by infection of SF9 insect cells cultured in SF-900 II medium (Invitrogen, Paisley, Scotland) with a baculovirus containing f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313752(US10167282, Compound TBAP-03)
Affinity DataIC50: 130nMAssay Description:V600EBRAF was generated by infection of SF9 insect cells cultured in SF-900 II medium (Invitrogen, Paisley, Scotland) with a baculovirus containing f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313754(US10167282, Compound TBAP-05)
Affinity DataIC50: 390nMAssay Description:V600EBRAF was generated by infection of SF9 insect cells cultured in SF-900 II medium (Invitrogen, Paisley, Scotland) with a baculovirus containing f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase B-raf [416-766,V600E](Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313754(US10167282, Compound TBAP-05)
Affinity DataIC50: 450nMAssay Description:Mutant BRAF WM266.4 Cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313751(US10167282, Compound TBAP-02)
Affinity DataIC50: 6.50E+4nMAssay Description:Studies were conducted at Cyprotex Discovery in Cheshire, UK according to the contractor's protocol. The studies were performed on an IonWorks HT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313750(US10167282, Compound TBAP-01)
Affinity DataIC50: 1.00E+5nMAssay Description:Studies were conducted at Cyprotex Discovery in Cheshire, UK according to the contractor's protocol. The studies were performed on an IonWorks HT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313752(US10167282, Compound TBAP-03)
Affinity DataIC50: 1.00E+5nMAssay Description:Studies were conducted at Cyprotex Discovery in Cheshire, UK according to the contractor's protocol. The studies were performed on an IonWorks HT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Cancer Research Technology

US Patent
LigandPNGBDBM313753(US10167282, Compound TBAP-04)
Affinity DataIC50: 1.00E+5nMAssay Description:Studies were conducted at Cyprotex Discovery in Cheshire, UK according to the contractor's protocol. The studies were performed on an IonWorks HT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2019
Entry Details
Go to US Patent