Compile Data Set for Download or QSAR
Report error Found 390 Enz. Inhib. hit(s) with all data for entry = 1119
TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310222(BDBM310223 | US10150760, Example 2.0 | (2S,3R)-N-(...)
Affinity DataEC50:  240nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310222(BDBM310223 | US10150760, Example 2.0 | (2S,3R)-N-(...)
Affinity DataEC50:  1.20E+3nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310224(US10150760, Example 4.0 | US10150760, Example 5.0)
Affinity DataEC50:  890nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310224(US10150760, Example 4.0 | US10150760, Example 5.0)
Affinity DataEC50: >4.20E+3nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310226(US10150760, Example 6.0)
Affinity DataEC50:  400nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310227(US10150760, Example 9.0 | (R)-2-(4-chlorophenyl)-N...)
Affinity DataEC50:  210nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310228(US10150760, Example 15.0 | US10150760, Example 17....)
Affinity DataEC50:  470nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310228(US10150760, Example 15.0 | US10150760, Example 17....)
Affinity DataEC50:  380nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310228(US10150760, Example 15.0 | US10150760, Example 17....)
Affinity DataEC50:  810nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310231(US10150760, Example 18.0)
Affinity DataEC50:  120nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310232(US10150760, Example 19.0)
Affinity DataEC50:  60nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310233(US10150760, Example 20.0 | US10150760, Example 21....)
Affinity DataEC50:  160nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310233(US10150760, Example 20.0 | US10150760, Example 21....)
Affinity DataEC50:  110nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310235(US10150760, Example 22.0 | US10150760, Example 23....)
Affinity DataEC50:  260nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310235(US10150760, Example 22.0 | US10150760, Example 23....)
Affinity DataEC50:  110nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310237(US10150760, Example 24.0 | (2S,3R)-3-(5-cyano-2-py...)
Affinity DataEC50:  4.5nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310238(US10150760, Example 25.0)
Affinity DataEC50:  130nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310239(US10150760, Example 26.0)
Affinity DataEC50:  870nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310240(US10150760, Example 35.0 | (2S,3R)-3-(5-chloro-2-p...)
Affinity DataEC50:  730nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310241(US10150760, Example 36.0)
Affinity DataEC50:  140nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310242(US10150760, Example 37.0)
Affinity DataEC50:  12nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310243(US10150760, Example 38.0)
Affinity DataEC50:  19nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310244(US10150760, Example 39.0)
Affinity DataEC50:  5.30nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310245(US10150760, Example 40.0)
Affinity DataEC50:  14nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310246(US10150760, Example 41.0)
Affinity DataEC50:  820nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310247(US10150760, Example 42.0)
Affinity DataEC50:  210nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310248(US10150760, Example 43.0 | 2-(2-cyano-4-fluorophen...)
Affinity DataEC50:  1.19E+3nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310249(US10150760, Example 44.0 | 2-(2-cyano-4-fluorophen...)
Affinity DataEC50:  430nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310250(US10150760, Example 45.0 | Preparation (1R,2S)-N-(...)
Affinity DataEC50:  510nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
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TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310251(US10150760, Example 47.0 | US10150760, Example 53....)
Affinity DataEC50:  0.720nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310252(US10150760, Example 48.0 | US10150760, Example 49....)
Affinity DataEC50:  3.90nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310252(US10150760, Example 48.0 | US10150760, Example 49....)
Affinity DataEC50:  1.80nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310252(US10150760, Example 48.0 | US10150760, Example 49....)
Affinity DataEC50:  28nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310255(US10150760, Example 51.0 | US10150760, Example 52....)
Affinity DataEC50:  0.590nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310255(US10150760, Example 51.0 | US10150760, Example 52....)
Affinity DataEC50:  20nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310251(US10150760, Example 47.0 | US10150760, Example 53....)
Affinity DataEC50:  13nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310258(US10150760, Example 54.0 | US10150760, Example 55....)
Affinity DataEC50:  37nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310258(US10150760, Example 54.0 | US10150760, Example 55....)
Affinity DataEC50:  66nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310260(US10150760, Example 56.0 | US10150760, Example 57....)
Affinity DataEC50:  19nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310260(US10150760, Example 56.0 | US10150760, Example 57....)
Affinity DataEC50:  21nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310262(US10150760, Example 58.0 | US10150760, Example 59....)
Affinity DataEC50:  120nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310262(US10150760, Example 58.0 | US10150760, Example 59....)
Affinity DataEC50:  16nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310264(US10150760, Example 60.0 | US10150760, Example 61....)
Affinity DataEC50:  9.30nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310264(US10150760, Example 60.0 | US10150760, Example 61....)
Affinity DataEC50:  29nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310266(US10150760, Example 62.0 | US10150760, Example 63....)
Affinity DataEC50:  26nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310266(US10150760, Example 62.0 | US10150760, Example 63....)
Affinity DataEC50:  1.5nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310268(US10150760, Example 64.0 | US10150760, Example 65....)
Affinity DataEC50:  29nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310268(US10150760, Example 64.0 | US10150760, Example 65....)
Affinity DataEC50:  2.90nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310270(US10150760, Example 66.0 | US10150760, Example 67....)
Affinity DataEC50:  6.90nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310270(US10150760, Example 66.0 | US10150760, Example 67....)
Affinity DataEC50:  180nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

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