Compile Data Set for Download or QSAR
Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 978
TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301696(US10131692, Compound 28)
Affinity DataEC50: >1.00E+7nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301701(US10131692, Compound 33)
Affinity DataEC50:  1.60E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301701(US10131692, Compound 33)
Affinity DataEC50:  100nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301700(US10131692, Compound 32)
Affinity DataEC50:  1.50E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301700(US10131692, Compound 32)
Affinity DataEC50:  290nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301699(US10131692, Compound 31)
Affinity DataEC50:  2.58E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301699(US10131692, Compound 31)
Affinity DataEC50:  100nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301698(US10131692, Compound 30)
Affinity DataEC50:  1.23E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301698(US10131692, Compound 30)
Affinity DataEC50:  190nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301697(US10131692, Compound 29)
Affinity DataEC50: >1.00E+7nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301697(US10131692, Compound 29)
Affinity DataEC50:  380nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301702(US10131692, Compound 34)
Affinity DataEC50:  110nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301696(US10131692, Compound 28)
Affinity DataEC50:  320nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301684(US10131692, Compound 27 | US10131692, Compound 16)
Affinity DataEC50:  1.33E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301684(US10131692, Compound 27 | US10131692, Compound 16)
Affinity DataEC50:  200nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301694(US10131692, Compound 26)
Affinity DataEC50:  4.58E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301694(US10131692, Compound 26)
Affinity DataEC50:  270nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301693(US10131692, Compound 25)
Affinity DataEC50:  6.43E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301693(US10131692, Compound 25)
Affinity DataEC50:  80nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301692(US10131692, Compound 24)
Affinity DataEC50:  2.23E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301692(US10131692, Compound 24)
Affinity DataEC50:  350nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301691(US10131692, Compound 23)
Affinity DataEC50:  5.18E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301707(US10131692, Compound 39)
Affinity DataEC50:  3.29E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataEC50:  5.40E+3nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataEC50:  40nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301711(US10131692, Compound 43 ([Val4]dDAVP))
Affinity DataEC50:  2.41E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301711(US10131692, Compound 43 ([Val4]dDAVP))
Affinity DataEC50:  50nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM50205308(CHEMBL1429 | (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino...)
Affinity DataEC50:  6.59E+3nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM50205308(CHEMBL1429 | (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino...)
Affinity DataEC50:  220nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301709(US10131692, Compound 41)
Affinity DataEC50:  1.14E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301709(US10131692, Compound 41)
Affinity DataEC50:  220nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
Go to US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301708(US10131692, Compound 40)
Affinity DataEC50:  1.41E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
Go to US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301708(US10131692, Compound 40)
Affinity DataEC50:  120nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301691(US10131692, Compound 23)
Affinity DataEC50:  100nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301707(US10131692, Compound 39)
Affinity DataEC50:  310nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301706(US10131692, Compound 38)
Affinity DataEC50:  1.50E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
Go to US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301706(US10131692, Compound 38)
Affinity DataEC50:  260nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
Go to US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301705(US10131692, Compound 37)
Affinity DataEC50:  1.01E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
Go to US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301705(US10131692, Compound 37)
Affinity DataEC50:  300nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
Go to US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301704(US10131692, Compound 36)
Affinity DataEC50:  9.56E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
Go to US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301704(US10131692, Compound 36)
Affinity DataEC50:  170nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301703(US10131692, Compound 35)
Affinity DataEC50:  1.22E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301703(US10131692, Compound 35)
Affinity DataEC50:  210nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301702(US10131692, Compound 34)
Affinity DataEC50:  4.02E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301674(US10131692, Compound 6)
Affinity DataEC50:  5.76E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301679(US10131692, Compound 11)
Affinity DataEC50:  4.80E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301679(US10131692, Compound 11)
Affinity DataEC50:  230nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301678(US10131692, Compound 10)
Affinity DataEC50:  1.05E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
Go to US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandPNGBDBM301678(US10131692, Compound 10)
Affinity DataEC50:  70nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301677(US10131692, Compound 9)
Affinity DataEC50: >1.00E+7nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
Go to US Patent

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