Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 824
TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandPNGBDBM293397(US10106522, Example 1)
Affinity DataIC50: 25nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
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Date in BDB:
2/24/2019
Entry Details
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TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandPNGBDBM293403(US10106522, Example 3)
Affinity DataIC50: 28nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
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Date in BDB:
2/24/2019
Entry Details
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TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandPNGBDBM293407(US10106522, Example 5)
Affinity DataIC50: 54nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
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Date in BDB:
2/24/2019
Entry Details
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TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandPNGBDBM293406(US10106522, Example 4)
Affinity DataIC50: 93nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
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Date in BDB:
2/24/2019
Entry Details
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TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandPNGBDBM293400(US10106522, Example 2)
Affinity DataIC50: 115nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
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Date in BDB:
2/24/2019
Entry Details
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TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandPNGBDBM293409(US10106522, Example 8)
Affinity DataIC50: 169nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
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Date in BDB:
2/24/2019
Entry Details
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TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandPNGBDBM293408(US10106522, Example 7)
Affinity DataIC50: 175nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
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Date in BDB:
2/24/2019
Entry Details
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TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandPNGBDBM293410(US10106522, Example 9)
Affinity DataIC50: 195nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
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Date in BDB:
2/24/2019
Entry Details
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TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandPNGBDBM293414(US10106522, Compound I-11 in CN 103896915)
Affinity DataIC50: 260nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
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Date in BDB:
2/24/2019
Entry Details
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TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandPNGBDBM293413(US10106522, Compound I-3 in CN 103896915)
Affinity DataIC50: 271nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
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Date in BDB:
2/24/2019
Entry Details
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TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandPNGBDBM293411(US10106522, Example 5 in EP 0580541)
Affinity DataIC50: 424nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
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Date in BDB:
2/24/2019
Entry Details
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TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandPNGBDBM293412(US10106522, Compound I-8 in CN 103896915)
Affinity DataIC50: 1.99E+3nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
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