Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 748
TargetGhrelin O-acyltransferase(Human)
Eli Lilly

US Patent
LigandPNGBDBM289087(US10093651, Example 15 | N-[(1S)-2-[4-[2-[4-Amino-...)
Affinity DataIC50: 55.7nMpH: 7.5Assay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO to obtain a ten-point dilution curve wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
Go to US Patent

TargetGhrelin O-acyltransferase(Human)
Eli Lilly

US Patent
LigandPNGBDBM289086(US10093651, Example 2 | N-[(1 S)-2-[4-[2-[4-Amino-...)
Affinity DataIC50: 69.5nMpH: 7.5Assay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO to obtain a ten-point dilution curve wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
Go to US Patent

TargetGhrelin O-acyltransferase(Human)
Eli Lilly

US Patent
LigandPNGBDBM289089(US10093651, Example 18 | N-[(1S)-2-[4-[2-[4-Amino-...)
Affinity DataIC50: 276nMpH: 7.5Assay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO to obtain a ten-point dilution curve wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
Go to US Patent

TargetGhrelin O-acyltransferase(Human)
Eli Lilly

US Patent
LigandPNGBDBM289088(US10093651, Example 17 | N-[(1S)-2-[4-[2-[4-Amino-...)
Affinity DataIC50: 420nMpH: 7.5Assay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO to obtain a ten-point dilution curve wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
Go to US Patent

TargetGhrelin O-acyltransferase(Human)
Eli Lilly

US Patent
LigandPNGBDBM289090(US10093651, Example 20 | Methyl-[(1S)-2-[4-[2-[4-a...)
Affinity DataIC50: 615nMpH: 7.5Assay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO to obtain a ten-point dilution curve wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
Go to US Patent