Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 3497
TargetVascular endothelial growth factor receptor 2(Human)
Allergan

US Patent
LigandPNGBDBM308058(US9650366, 9 | US10011593, Ex. 9)
Affinity DataIC50: 5nMAssay Description:VEGFR2: Biochemical KDR kinase assays were performed in 96 well microtiter plates that were coated overnight with 75 μg/well of poly-Glu-Tyr (4:...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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TargetVascular endothelial growth factor receptor 2(Human)
Allergan

US Patent
LigandPNGBDBM308059(US9650366, 10 | US10011593, Ex. 10)
Affinity DataIC50: 7nMAssay Description:VEGFR2: Biochemical KDR kinase assays were performed in 96 well microtiter plates that were coated overnight with 75 μg/well of poly-Glu-Tyr (4:...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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TargetVascular endothelial growth factor receptor 2(Human)
Allergan

US Patent
LigandPNGBDBM308061(US9650366, 12 | US10011593, Ex. 12)
Affinity DataIC50: 8nMAssay Description:VEGFR2: Biochemical KDR kinase assays were performed in 96 well microtiter plates that were coated overnight with 75 μg/well of poly-Glu-Tyr (4:...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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TargetPlatelet-derived growth factor receptor beta(Human)
Allergan

US Patent
LigandPNGBDBM308058(US9650366, 9 | US10011593, Ex. 9)
Affinity DataIC50: 21nMAssay Description:PDGFRβ: Biochemical PDGFRβ kinase assays were performed in 96 well microtiter plates that were coated overnight with 75 μg of poly-Glu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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LigandPNGBDBM308051(US9650366, 3 | US10011593, Ex. 3)
Affinity DataIC50: 39nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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LigandPNGBDBM308056(US9650366, 6 | US10011593, Ex. 6)
Affinity DataIC50: 66nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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LigandPNGBDBM308055(US9650366, 5 | US10011593, Ex. 5)
Affinity DataIC50: 76nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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LigandPNGBDBM308057(US9650366, 8 | US10011593, Ex. 8)
Affinity DataIC50: 82nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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LigandPNGBDBM308054(US9650366, 4 | US10011593, Ex. 4)
Affinity DataIC50: 99nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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LigandPNGBDBM308050(US9650366, 2 | US10011593, Ex. 2)
Affinity DataIC50: 140nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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LigandPNGBDBM308060(US9650366, 11 | US10011593, Ex. 11)
Affinity DataIC50: 158nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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LigandPNGBDBM308063(US9650366, 14 | US10011593, Ex. 14)
Affinity DataIC50: 301nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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LigandPNGBDBM308062(US9650366, 13 | US10011593, Ex. 13)
Affinity DataIC50: 558nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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LigandPNGBDBM308049(US9650366, 1 | US10011593, Ex. 1)
Affinity DataIC50: 727nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
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LigandPNGBDBM308058(US9650366, 9 | US10011593, Ex. 9)
Affinity DataIC50: 1.00E+4nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
Go to US Patent

LigandPNGBDBM308061(US9650366, 12 | US10011593, Ex. 12)
Affinity DataIC50: 1.00E+4nMAssay Description:PKR: Commercially available recombinant human GST-PKR (SignalChem, Canada; 1.5 uM-2 uM stock) is diluted to 500 nM in assay buffer (20 mM Tris-HCl, p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
Go to US Patent