Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50008263
TargetD(3) dopamine receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071958(Biphenylene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi:  0.900nMAssay Description:Compound was evaluated for binding affinity against human Dopamine receptor D3 transfected in CHO cell membranes to stimulate [3H]thymidine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071959(9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi:  1.40nMAssay Description:Compound was evaluated for binding affinity against human Dopamine receptor D3 transfected in CHO cell membranes to stimulate [3H]thymidine uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071960(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  65nMAssay Description:Affinity against D4 receptor was evaluatedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071958(Biphenylene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi:  125nMAssay Description:Compound was evaluated for binding affinity against 5-hydroxytryptamine 2 receptor from ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071959(9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi:  217nMAssay Description:Compound was evaluated for binding affinity against Dopamine receptor D2 subtype from primateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071959(9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi:  223nMAssay Description:Compound was evaluated for binding affinity against 5-hydroxytryptamine 2 receptor from ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071958(Biphenylene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi:  262nMAssay Description:Compound was evaluated for binding affinity against Dopamine receptor D2 subtype from primateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50071958(Biphenylene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi:  547nMAssay Description:Compound was evaluated for binding affinity against Alpha-1 adrenergic receptor from ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50071959(9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi:  642nMAssay Description:Compound was evaluated for binding affinity against Alpha-1 adrenergic receptor from ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071958(Biphenylene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi: >5.00E+3nMAssay Description:Compound was evaluated for binding affinity against human Dopamine receptor D4 transfected in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071959(9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi: >5.00E+3nMAssay Description:Compound was evaluated for binding affinity against human Dopamine receptor D4 transfected in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071958(Biphenylene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for binding affinity against Dopamine receptor D1 transfected in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1B) dopamine receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071958(Biphenylene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for binding affinity against human Dopamine receptor D5 transfected in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1B) dopamine receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071959(9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for binding affinity against human Dopamine receptor D5 transfected in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50071959(9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for binding affinity against Dopamine receptor D1 transfected in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed