Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50034984
TargetDelta-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  0.217nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  27nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  30nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50291697((1S,2S,13S)-22-(cyclopropylmethyl)-14-oxa-11,22-di...)
Affinity DataKi:  35nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069179(22-cyclopropylmethyl-16-vinyl-14-oxa-11,22-diazahe...)
Affinity DataKi:  61nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069175(22-cyclopropylmethyl-16-methyl-14-oxa-11,22-diazah...)
Affinity DataKi:  71nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069177(22-cyclopropylmethyl-16-(2-furyl)-14-oxa-11,22-dia...)
Affinity DataKi:  959nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069176(22-cyclopropylmethyl-16-(3-hydroxyphenyl)-14-oxa-1...)
Affinity DataKi:  1.61E+3nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069179(22-cyclopropylmethyl-16-vinyl-14-oxa-11,22-diazahe...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069177(22-cyclopropylmethyl-16-(2-furyl)-14-oxa-11,22-dia...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069180(22-cyclopropylmethyl-16-(3-methoxyphenyl)-14-oxa-1...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069181(22-cyclopropylmethyl-16-phenyl-14-oxa-11,22-diazah...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50291697((1S,2S,13S)-22-(cyclopropylmethyl)-14-oxa-11,22-di...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069175(22-cyclopropylmethyl-16-methyl-14-oxa-11,22-diazah...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069176(22-cyclopropylmethyl-16-(3-hydroxyphenyl)-14-oxa-1...)
Affinity DataKi: >5.68E+3nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069180(22-cyclopropylmethyl-16-(3-methoxyphenyl)-14-oxa-1...)
Affinity DataKi: >6.67E+3nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069177(22-cyclopropylmethyl-16-(2-furyl)-14-oxa-11,22-dia...)
Affinity DataKi: >6.80E+3nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069181(22-cyclopropylmethyl-16-phenyl-14-oxa-11,22-diazah...)
Affinity DataKi: >6.80E+3nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069176(22-cyclopropylmethyl-16-(3-hydroxyphenyl)-14-oxa-1...)
Affinity DataKi: >6.80E+3nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069180(22-cyclopropylmethyl-16-(3-methoxyphenyl)-14-oxa-1...)
Affinity DataKi: >6.80E+3nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069175(22-cyclopropylmethyl-16-methyl-14-oxa-11,22-diazah...)
Affinity DataKi: >6.80E+3nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069181(22-cyclopropylmethyl-16-phenyl-14-oxa-11,22-diazah...)
Affinity DataKi:  1.06E+4nMAssay Description:Compound was tested for its ability to displace [3H]DADLE from delta receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50291697((1S,2S,13S)-22-(cyclopropylmethyl)-14-oxa-11,22-di...)
Affinity DataKi:  1.09E+4nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50069179(22-cyclopropylmethyl-16-vinyl-14-oxa-11,22-diazahe...)
Affinity DataKi:  1.76E+4nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from kappa receptor in guinea pig brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed