Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50007888
TargetLactoylglutathione lyase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50069024(2-Amino-4-[1-(carboxymethyl-carbamoyl)-3-(hydroxy-...)
Affinity DataKi:  1.90E+3nMAssay Description:Compound was evaluated for inhibition of Saccharomyces cerevisiae glyoxalase-I by using enzymatic assay at each of 6 substrate concentrations between...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLactoylglutathione lyase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50069024(2-Amino-4-[1-(carboxymethyl-carbamoyl)-3-(hydroxy-...)
Affinity DataIC50: 3.90E+3nMAssay Description:Compound was evaluated for inhibition of Saccharomyces cerevisiae glyoxalase-I, activity is determined with 0.5 mM substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLactoylglutathione lyase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50241121(S-p-bromobenzyl glutatione | S-p-bromobenzylglutat...)
Affinity DataKi:  4.30E+3nMAssay Description:Compound was evaluated for inhibition of Saccharomyces cerevisiae glyoxalase-I by using enzymatic assay at each of 6 substrate concentrations between...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLactoylglutathione lyase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50241121(S-p-bromobenzyl glutatione | S-p-bromobenzylglutat...)
Affinity DataIC50: 8.20E+3nMAssay Description:Compound was evaluated for inhibition of Saccharomyces cerevisiae glyoxalase-I, activity i determined with 0.5 mM substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLactoylglutathione lyase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50069025(2-Amino-4-[1-(carboxymethyl-carbamoyl)-3-hydroxyca...)
Affinity DataKi:  9.29E+4nMAssay Description:Compound was evaluated for inhibition of Saccharomyces cerevisiae glyoxalase-I by using enzymatic assay at each of 6 substrate concentrations between...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLactoylglutathione lyase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50069026(2-Amino-4-[1-(ethoxycarbonylmethyl-carbamoyl)-3-(h...)
Affinity DataIC50: 1.41E+5nMAssay Description:Compound was evaluated for inhibition of Saccharomyces cerevisiae glyoxalase-I, activity is determined with 0.5 mM substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLactoylglutathione lyase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50069025(2-Amino-4-[1-(carboxymethyl-carbamoyl)-3-hydroxyca...)
Affinity DataIC50: 2.10E+5nMAssay Description:Compound was evaluated for inhibition of Saccharomyces cerevisiae glyoxalase-I, activity is determined with 0.5 mM substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLactoylglutathione lyase(Human)
University of Waterloo

Curated by ChEMBL
LigandPNGBDBM50069027(2-Amino-4-[1-(ethoxycarbonylmethyl-carbamoyl)-3-hy...)
Affinity DataIC50: 1.62E+6nMAssay Description:Compound was evaluated for inhibition of Saccharomyces cerevisiae glyoxalase-I, activity is determined with 0.5 mM substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed