Compile Data Set for Download or QSAR
Report error Found 67 Enz. Inhib. hit(s) with all data for entry = 50036606
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062005(PD-135666 | 3-[2-(2-Adamantan-2-yl-acetylamino)-3-...)
Affinity DataIC50: 0.150nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062000(2-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-in...)
Affinity DataIC50: 0.990nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50449787(PD-134308 | CHEMBL2062154)
Affinity DataIC50: 1.70nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062003([(R)-2-(1H-Indol-3-yl)-1-((R)-2-methoxymethyl-pyrr...)
Affinity DataIC50: 2.5nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061997([(R)-1-((1R,2R)-2-Hydroxy-cyclohexylcarbamoyl)-2-(...)
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061994([(R)-1-(2-Cyano-cyclohexylcarbamoyl)-2-(1H-indol-3...)
Affinity DataIC50: 3.5nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062006([(R)-1-((1R,2R)-2-Hydroxy-cycloheptylcarbamoyl)-2-...)
Affinity DataIC50: 4.70nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062001([(R)-1-(2-Hydroxy-cyclohexylcarbamoyl)-2-(1H-indol...)
Affinity DataIC50: 6.20nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061988([(R)-1-((S)-1-Hydroxymethyl-2-phenyl-ethylcarbamoy...)
Affinity DataIC50: 6.30nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061993([(R)-1-(3-Aza-bicyclo[3.2.2]non-3-ylcarbamoyl)-2-(...)
Affinity DataIC50: 6.5nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061990((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 9.30nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062008([(R)-1-(Azepan-1-ylcarbamoyl)-2-(1H-indol-3-yl)-1-...)
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50454908(CHEMBL2112795)
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062012([(R)-2-(1H-Indol-3-yl)-1-methyl-1-(piperidin-1-ylc...)
Affinity DataIC50: 20nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061999([(R)-1-(1-Benzyl-2-phenyl-ethylcarbamoyl)-2-(1H-in...)
Affinity DataIC50: 20nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062005(PD-135666 | 3-[2-(2-Adamantan-2-yl-acetylamino)-3-...)
Affinity DataIC50: 26nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062015([(R)-1-((1S,2S)-2-Hydroxy-cycloheptylcarbamoyl)-2-...)
Affinity DataIC50: 26nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50366633(CHEMBL1169566)
Affinity DataIC50: 32nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062004([(R)-2-(1H-Indol-3-yl)-1-methyl-1-(2-methyl-cycloh...)
Affinity DataIC50: 39nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50006875(N-{(S)-2-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3...)
Affinity DataIC50: 43nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061998([(R)-1-Cycloheptylcarbamoyl-2-(1H-indol-3-yl)-1-me...)
Affinity DataIC50: 46nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50366633(CHEMBL1169566)
Affinity DataIC50: 48nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061995([(R)-1-Cyclohexylcarbamoyl-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50: 50nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062014([(R)-2-(1H-Indol-3-yl)-1-((S)-2-methoxymethyl-pyrr...)
Affinity DataIC50: 65nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062013([(R)-1-(Bicyclo[2.2.1]hept-2-ylcarbamoyl)-2-(1H-in...)
Affinity DataIC50: 78.5nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062013([(R)-1-(Bicyclo[2.2.1]hept-2-ylcarbamoyl)-2-(1H-in...)
Affinity DataIC50: 79nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062018(1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-in...)
Affinity DataIC50: 83nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062016([(R)-1-(1-Hydroxymethyl-cyclohexylcarbamoyl)-2-(1H...)
Affinity DataIC50: 121nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062009([(R)-2-(1H-Indol-3-yl)-1-methyl-1-(pyrrolidin-1-yl...)
Affinity DataIC50: 132nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061990((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 186nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061992(1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-in...)
Affinity DataIC50: 191nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062002(3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-in...)
Affinity DataIC50: 214nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062010([(R)-1-(1-Hydroxymethyl-cyclopentylcarbamoyl)-2-(1...)
Affinity DataIC50: 268nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061991([(R)-3-Cyclohexylamino-1-(1H-indol-3-ylmethyl)-1-m...)
Affinity DataIC50: 314nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062017([(R)-2-(1H-Indol-3-yl)-1-methyl-1-phenylcarbamoyl-...)
Affinity DataIC50: 327nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50366633(CHEMBL1169566)
Affinity DataIC50: 650nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50366633(CHEMBL1169566)
Affinity DataIC50: 650nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062000(2-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-in...)
Affinity DataIC50: 701nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061988([(R)-1-((S)-1-Hydroxymethyl-2-phenyl-ethylcarbamoy...)
Affinity DataIC50: 780nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062002(3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-in...)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062006([(R)-1-((1R,2R)-2-Hydroxy-cycloheptylcarbamoyl)-2-...)
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062001([(R)-1-(2-Hydroxy-cyclohexylcarbamoyl)-2-(1H-indol...)
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062010([(R)-1-(1-Hydroxymethyl-cyclopentylcarbamoyl)-2-(1...)
Affinity DataIC50: 1.42E+3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062013([(R)-1-(Bicyclo[2.2.1]hept-2-ylcarbamoyl)-2-(1H-in...)
Affinity DataIC50: 1.46E+3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062013([(R)-1-(Bicyclo[2.2.1]hept-2-ylcarbamoyl)-2-(1H-in...)
Affinity DataIC50: 1.46E+3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061994([(R)-1-(2-Cyano-cyclohexylcarbamoyl)-2-(1H-indol-3...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062016([(R)-1-(1-Hydroxymethyl-cyclohexylcarbamoyl)-2-(1H...)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062018(1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-in...)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50061993([(R)-1-(3-Aza-bicyclo[3.2.2]non-3-ylcarbamoyl)-2-(...)
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50062015([(R)-1-((1S,2S)-2-Hydroxy-cycloheptylcarbamoyl)-2-...)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
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