Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50004753
TargetSolute carrier family 15 member 2(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50370586(CEFTIBUTEN | 7-(2-(2-amino-4-thiazolyl)-4-carboxy-...)
Affinity DataKi:  9.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetSolute carrier family 15 member 2(Rat)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50370586(CEFTIBUTEN | 7-(2-(2-amino-4-thiazolyl)-4-carboxy-...)
Affinity DataKi:  3.80E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in SKPT cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50370586(CEFTIBUTEN | 7-(2-(2-amino-4-thiazolyl)-4-carboxy-...)
Affinity DataKi:  7.10E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50370586(CEFTIBUTEN | 7-(2-(2-amino-4-thiazolyl)-4-carboxy-...)
Affinity DataKi:  8.70E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in Caco-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetSolute carrier family 15 member 2(Rat)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM84007(SMR001307271 | Cefiximum [Latin] | cid_5362065 | M...)
Affinity DataIC50: 3.20E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 5 uM) in SKPT cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetSolute carrier family 15 member 2(Rat)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50248190(CHEBI:3485 | CI-983 | Cefdinir | Cefzon | FK-482 |...)
Affinity DataIC50: 1.00E+7nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 5 uM) in SKPT cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM84007(SMR001307271 | Cefiximum [Latin] | cid_5362065 | M...)
Affinity DataIC50: 1.00E+7nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 5 uM) in Caco-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed