Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with all data for entry = 50036596
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056947(N-{2-[4-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-piper...)
Affinity DataIC50: 14nMAssay Description:Inhibition of forskolin-activated adenylate cyclase (cAMP) activity at 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataIC50: 14nMAssay Description:Inhibition of forskolin-activated adenylate cyclase (cAMP) activity at 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056945(4-Chloro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataIC50: 38nMAssay Description:Inhibition of forskolin-activated adenylate cyclase (cAMP) activity at 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataIC50: 52nMAssay Description:Inhibition of forskolin-activated adenylate cyclase (cAMP) activity at 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056945(4-Chloro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataIC50: 75nMAssay Description:Inhibition of forskolin-activated adenylate cyclase (cAMP) activity at 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056946(1-(4-Fluoro-phenyl)-4-[4-(1,2,3,4-tetrahydro-napht...)
Affinity DataIC50: 210nMAssay Description:Inhibition of forskolin-activated adenylate cyclase (cAMP) activity at 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056944(4-Fluoro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of forskolin-activated adenylate cyclase (cAMP) activity at 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056947(N-{2-[4-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-piper...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056947(N-{2-[4-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-piper...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056944(4-Fluoro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Bovine)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM69602(WB-4101 hydrochloride | N-(2,3-dihydro-1,4-benzodi...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity of compound towards Alpha-1 adrenergic receptor using [3H]prazosin 0.5 nM ligand in frontal cortex calf was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50334150(1-(1-(4,4-bis(4-fluorophenyl)butyl)piperidin-4-yl)...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity of compound towards Dopamine receptor D2 using [3H]raclopride (1.2 nM) ligand in striatum bovine was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity against human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM31005(MIANSERIN HYDROCHLORIDE | SMR000058472 | MLS000069...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity of compound towards 5-hydroxytryptamine 1C receptor using [3H]mesulergine (1.2 nM) ligand in choroid Plexus pig was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056945(4-Chloro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Human)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  8.60nMAssay Description:Binding affinity of compound towards 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT (0.5 nM) ligand in hippocampus + frontal bovine was determin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  9.30nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Human)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  15nMAssay Description:Binding affinity against human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056946(1-(4-Fluoro-phenyl)-4-[4-(1,2,3,4-tetrahydro-napht...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Bovine)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50026957((cis) 2-{4-[3-(2-Trifluoromethyl-thioxanthen-9-yli...)
Affinity DataKi:  18nMAssay Description:Binding affinity of compound towards Dopamine receptor D1 using [3H]SCH-23390 (0.5 nM) ligand in striatum bovine was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Bovine)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056946(1-(4-Fluoro-phenyl)-4-[4-(1,2,3,4-tetrahydro-napht...)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]prazosin binding to Alpha-1 adrenergic receptor in bovine frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056946(1-(4-Fluoro-phenyl)-4-[4-(1,2,3,4-tetrahydro-napht...)
Affinity DataKi:  30nMAssay Description:Inhibition of [3H]DTG binding to sigma receptor in rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B/3C/3D/3E(Human)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  33nMAssay Description:Binding affinity of compound towards 5-hydroxytryptamine 3 receptor using [3H]-BRL-43694 (1 nM) ligand in NG cells 108-15 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  38nMAssay Description:Binding affinity of compound towards sigma receptor using [3H]DTG (4 nM) ligand in hippocampus rat was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistamine H1 receptor(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056946(1-(4-Fluoro-phenyl)-4-[4-(1,2,3,4-tetrahydro-napht...)
Affinity DataKi:  42nMAssay Description:Inhibition of [3H]pyrilamine binding to Histamine H1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  44nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2 of bovine striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  48nMAssay Description:Inhibition of [3H]DTG binding to sigma receptor in rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056944(4-Fluoro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056944(4-Fluoro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataKi:  58nMAssay Description:Inhibition of [3H]pyrilamine binding to Histamine H1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056944(4-Fluoro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataKi:  58nMAssay Description:Inhibition of [3H]pyrilamine binding to Histamine H1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056947(N-{2-[4-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-piper...)
Affinity DataKi:  70nMAssay Description:Inhibition of [3H]pyrilamine binding to Histamine H1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056947(N-{2-[4-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-piper...)
Affinity DataKi:  70nMAssay Description:Inhibition of [3H]pyrilamine binding to Histamine H1 receptor in rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  84nMAssay Description:Binding affinity against Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056947(N-{2-[4-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-piper...)
Affinity DataKi:  90nMAssay Description:Inhibition of [3H]DTG binding to sigma receptor in rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056946(1-(4-Fluoro-phenyl)-4-[4-(1,2,3,4-tetrahydro-napht...)
Affinity DataKi:  110nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2 of bovine striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  115nMAssay Description:Binding affinity of compound towards Dopamine receptor D3 using [3H]spiperone (1.2 nM) ligand in cortex was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056945(4-Chloro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataKi:  120nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2 of bovine striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056944(4-Fluoro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataKi:  130nMAssay Description:Inhibition of [3H]DTG binding to sigma receptor in rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056947(N-{2-[4-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-piper...)
Affinity DataKi:  130nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2 of bovine striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056947(N-{2-[4-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-piper...)
Affinity DataKi:  130nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2 of bovine striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Bovine)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  178nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056944(4-Fluoro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataKi:  190nMAssay Description:Inhibition of [3H]DTG binding to sigma receptor in rat hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056945(4-Chloro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataKi:  480nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2 of bovine striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056945(4-Chloro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataKi:  650nMAssay Description:Inhibition of [3H]mesulergine binding to 5-hydroxytryptamine 1C receptor of pig choroid PlexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056945(4-Chloro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataKi:  650nMAssay Description:Inhibition of [3H]mesulergine binding to 5-hydroxytryptamine 1C receptor of pig choroid PlexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  660nMAssay Description:Inhibition of [3H]spiperone binding to Dopamine receptor D3 in bovine cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
Cooperation Pharmaceutique Fran�Aise

Curated by ChEMBL
LigandPNGBDBM50056944(4-Fluoro-N-{2-[4-(1,2,3,4-tetrahydro-naphthalen-1-...)
Affinity DataKi:  740nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2 of bovine striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
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