Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50006962
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM7585(2,6,9-Trisubstituted purine deriv. 27 | CHEMBL5238...)
Affinity DataIC50: 650nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056163((S)-2-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamin...)
Affinity DataIC50: 800nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056169(1-(6-Benzylamino-9-isopropyl-9H-purin-2-ylamino)-p...)
Affinity DataIC50: 900nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM10636(6-(benzylamino)-2-[(2-hydroxyethyl)amino]-9-isopro...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056159(2-[6-(Cyclohexyl-methyl-amino)-9-methyl-9H-purin-2...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM5718(2,6,9-Trisubstituted purine deriv. 26 | 2-{[6-(ben...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056177(2-[6-Benzylamino-2-(2-hydroxy-ethylamino)-purin-9-...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056174(Benzyl-(2-chloro-9-methyl-9H-purin-6-yl)-amine | C...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056168(Benzyl-(2-chloro-9-isopropyl-9H-purin-6-yl)-amine ...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056164(2-(6-Benzylamino-9H-purin-2-ylamino)-ethanol | CHE...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056160(Benzyl-(9-methyl-9H-purin-6-yl)-amine | CHEMBL1310...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056176((2-Chloro-9-methyl-9H-purin-6-yl)-(3-methyl-but-2-...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056170(N*6*-Benzyl-9-methyl-9H-purine-2,6-diamine | CHEMB...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056172(2-(6-Amino-9-methyl-9H-purin-2-ylamino)-ethanol | ...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056165(2-[9-Methyl-6-(3-methyl-but-2-enylamino)-9H-purin-...)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50009702(CHEMBL317398 | 2-Chloro-9-methyl-9H-purin-6-ylamin...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056167(N*6*-Benzyl-9H-purine-2,6-diamine | CHEMBL133214)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50208879(9H-Purine-2,6-diamine0.5M H2SO4 | 2,6-diaminopurin...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of purified Cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis (precipitation at the higher concentra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056173((2-Chloro-9-methyl-9H-purin-6-yl)-cyclohexyl-methy...)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50205363(N-benzyl-9H-purin-6-amine | N-benzyladenine | 6-(b...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM33218(CHEMBL226345 | Adenine, 1 | purine, 6)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056161(2-(6-Amino-9H-purin-2-ylamino)-ethanol | CHEMBL130...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056162(Benzyl-(3-methyl-3,9-dihydro-2H-purin-6-yl)-amine ...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50030961(2-Methyl-9H-purin-6-ylamine | CHEMBL330897)
Affinity DataIC50: 3.20E+5nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50009685(CHEMBL65976 | 9-Methyl-9H-purin-6-ylamine | 9-Meth...)
Affinity DataIC50: 3.50E+5nMAssay Description:Inhibition of purified Cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis (precipitation at the higher concentra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056171(3-Methyl-3,9-dihydro-2H-purin-6-ylamine | CHEMBL13...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056175(7-Methyl-8,9-dihydro-7H-purin-6-ylamine | CHEMBL33...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056166(1-Methyl-6,9-dihydro-1H-purin-6-ylamine | 1-Methyl...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056179(Benzyl-(7-methyl-8,9-dihydro-7H-purin-6-yl)-amine ...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056180(2-Chloro-9H-purin-6-ylamine | CHEMBL134192 | EN300...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of purified Cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis (precipitation at the higher concentra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Charles University

Curated by ChEMBL
LigandPNGBDBM50056181(Benzyl-(1-methyl-6,9-dihydro-1H-purin-6-yl)-amine ...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against purified cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed