Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 50041249
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408031(Ro-20-1815 | CHEMBL151121)
Affinity DataIC50: 1.53E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408022(Ro-07-4419 | CHEMBL151386)
Affinity DataIC50: 5.26E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408023(Ro-20-8895 | CHEMBL346213)
Affinity DataIC50: 5.26E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50026859(7-Chloro-5-(2,6-dichloro-phenyl)-1-methyl-1,3-dihy...)
Affinity DataIC50: 1.81E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50040701(Ro-22-6762 | 7,8-Dichloro-1-methyl-5-phenyl-1,3-di...)
Affinity DataIC50: 2.50E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408024(Ro-05-2904 | RO-052904)
Affinity DataIC50: 7.69E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408025(Ro-20-3053 | CHEMBL151179)
Affinity DataIC50: 5.55E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408026(Ro-05-4336 | CHEMBL147024)
Affinity DataIC50: 4.76E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50292627(Lorazepam preservative free | (RS)-9-chloro-6-(2-c...)
Affinity DataIC50: 2.85E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408027(Ro-05-3590 | CHEMBL314775)
Affinity DataIC50: 2.85E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50020856(7-nitro-5-phenyl-1H-benzo[e][1,4]diazepin-2(3H)-on...)
Affinity DataIC50: 9.99E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408028(Ro-05-6820 | CHEMBL151984)
Affinity DataIC50: 1.35E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50026855(7-Chloro-5-(2,6-dichloro-phenyl)-1,3-dihydro-benzo...)
Affinity DataIC50: 1.42E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408029(Ro-14-3074 | CHEMBL341902)
Affinity DataIC50: 1.88E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408030(CHEMBL345301)
Affinity DataIC50: 1.42E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM25878(Flunitrazepam | [3H]Rohypnol | 5-(2-fluorophenyl)-...)
Affinity DataIC50: 2.63E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataIC50: 1.23E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408032(Restoril | Temaz | TEMAZEPAM)
Affinity DataIC50: 6.25E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50027835(CHEMBL523 | Nordazepam | Gen-Xene | 7-chloro-5-phe...)
Affinity DataIC50: 1.06E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408033(Ro-20-5397 | CHEMBL348694)
Affinity DataIC50: 2.32E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408034(Ro-20-7078 | CHEMBL148490)
Affinity DataIC50: 1.88E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408035(Ro-05-4435 | CHEMBL87369)
Affinity DataIC50: 6.66E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50026858(CHEMBL268254 | 7-chloro-5-(2-chlorophenyl)-1H-benz...)
Affinity DataIC50: 5.55E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408036(7-Aminoclonazepam | Ro-05-4619 | CHEMBL1273)
Affinity DataIC50: 1.33E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408037(CHEMBL149268)
Affinity DataIC50: 8.33E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408038(Ro-05-4865 | CHEMBL150738)
Affinity DataIC50: 5.88E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408039(Ro-06-7263 | CHEMBL150925)
Affinity DataIC50: 2.04E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50040705(Ro-20-5747 | 5-Phenyl-7-vinyl-1,3-dihydro-benzo[e]...)
Affinity DataIC50: 4.16E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408040(Ro-05-4082 | RO-054082)
Affinity DataIC50: 4.54E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408012(CHEMBL150323)
Affinity DataIC50: 2.85E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50422186(Ro-05-3072 | CHEMBL147144)
Affinity DataIC50: 2.58E+6nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50422184(Ro-20-1310 | CHEMBL140487)
Affinity DataIC50: 1.61E+6nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50422187(Ro-05-3418 | CHEMBL150977)
Affinity DataIC50: 2.17E+6nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50083882(CHEMBL275115 | QHII-066 | 1-Methyl-2-oxo-5-phenyl-...)
Affinity DataIC50: 2.63E+6nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50422185(Ro-22-4683 | CHEMBL345284)
Affinity DataIC50: 3.33E+6nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50083899(5-Phenyl-1,3-dihydro-benzo[e][1,4]diazepin-2-one |...)
Affinity DataIC50: 2.85E+6nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408006(Ro-07-5193 | CHEMBL148526)
Affinity DataIC50: 3.33E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408007(Ro-20-7736 | CHEMBL358955)
Affinity DataIC50: 1.04E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50040702(Ro-20-8552 | 8-Chloro-5-(2-fluoro-phenyl)-7-methyl...)
Affinity DataIC50: 7.14E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408008(Ro-07-4065 | CHEMBL346673)
Affinity DataIC50: 2.43E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408009(Ro-07-2750 | CHEMBL435684)
Affinity DataIC50: 4.08E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408010(Ro-05-4608 | CHEMBL358422)
Affinity DataIC50: 2.63E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408011(Ro-07-3953 | CHEMBL151574)
Affinity DataIC50: 6.25E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50422188(Ro-06-9098 | MOTRAZEPAM)
Affinity DataIC50: 2.32E+6nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408013(Ro-07-6198 | CHEMBL151548)
Affinity DataIC50: 3.57E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408014(N-Desalkyl-2-Oxoquazepam | Ro-05-3367 | CHEMBL974)
Affinity DataIC50: 5.00E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408015(Ro-05-6822 | CHEMBL85481)
Affinity DataIC50: 1.95E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408016(Ro-05-3061 | RO-053061)
Affinity DataIC50: 2.50E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408017(Ro-07-9957 | CHEMBL358426)
Affinity DataIC50: 3.45E+8nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50408018(HALAZEPAM)
Affinity DataIC50: 1.08E+7nMAssay Description:Binding affinity of compound towards Benzodiazepine receptor in a competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
Displayed 1 to 50 (of 57 total ) | Next | Last >>
Jump to: