Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50036463
TargetD(2) dopamine receptor(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50366495(CHEMBL1255588 | (+)butaclamol)
Affinity DataKi:  0.300nMAssay Description:Binding affinity was tested on Dopamine receptor D2 using radioligand [3H]spiroperidolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054122(2-[4-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-butyl]-1...)
Affinity DataKi:  66nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054118(Dipropyl-[4-(1,2,3,4-tetrahydro-naphthalen-1-yl)-b...)
Affinity DataKi:  200nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054113(4-Benzyl-1-[4-(1,2,3,4-tetrahydro-naphthalen-1-yl)...)
Affinity DataKi:  285nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054112([4-(3,4-Dihydro-naphthalen-1-yl)-butyl]-dipropyl-a...)
Affinity DataKi:  357nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50368882(SK&F-10047 | SK-10047 | CHEMBL147585)
Affinity DataKi:  370nMAssay Description:Binding affinity of compound was tested on Phencyclidine binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054115(Dipropyl-[3-(1,2,3,4-tetrahydro-naphthalen-1-yl)-p...)
Affinity DataKi:  400nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054124(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataKi:  898nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054116(4-Benzyl-1-[3-(5-methoxy-1,2,3,4-tetrahydro-naphth...)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity of compound towards Dopamine receptor D2 was determined in rat striatal homogenate using [3H]- spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054121(3,3-Dimethyl-1-[4-(1,2,3,4-tetrahydro-naphthalen-1...)
Affinity DataKi: >1.43E+3nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054110(1-[4-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-butyl]-p...)
Affinity DataKi: >1.43E+3nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054120(1-[3-(1,2,3,4-Tetrahydro-naphthalen-1-yl)-propyl]-...)
Affinity DataKi: >1.43E+3nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054119(1-[3-(4,5,6,7-Tetrahydro-benzo[c]thiophen-4-yl)-pr...)
Affinity DataKi: >1.43E+3nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054117(1-(3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)...)
Affinity DataKi: >1.43E+3nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054111(3,3-Dimethyl-1-[3-(4,5,6,7-tetrahydro-benzo[c]thio...)
Affinity DataKi: >1.43E+3nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054123(1-[4-(3,4-Dihydro-naphthalen-1-yl)-butyl]-piperidi...)
Affinity DataKi: >1.43E+3nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054114(1-[3-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataKi: >1.43E+3nMAssay Description:Binding affinity was tested on 5-hydroxytryptamine 1A receptor using radioligand [3H]5-HT binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054114(1-[3-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataKi: >1.85E+3nMAssay Description:Binding affinity was tested on Dopamine receptor D2 using radioligand [3H]spiroperidolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054117(1-(3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)...)
Affinity DataKi: >1.85E+3nMAssay Description:Binding affinity was tested on Dopamine receptor D2 using radioligand [3H]spiroperidolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054121(3,3-Dimethyl-1-[4-(1,2,3,4-tetrahydro-naphthalen-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was tested on Dopamine receptor D2 using radioligand [3H]spiroperidolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50054124(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was tested on Dopamine receptor D2 using radioligand [3H]spiroperidolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed