Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50006782
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50053589((S)-3-Hydroxyphenylglycine | 3HPG | CHEMBL442347 |...)
Affinity DataEC50:  6.80E+4nMAssay Description:Effective concentration for half maximal stimulation of PI hydrolysis (mGluR1a)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50034501((S)-Amino-(3-oxo-2,3-dihydro-isoxazol-5-yl)-acetic...)
Affinity DataEC50:  6.00E+3nMAssay Description:Effective concentration for half maximal stimulation of PI hydrolysis (mGluR1a)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM17660(2-amino-3-(3,5-dioxo[1,2,4]oxadiazolidin-2-yl)prop...)
Affinity DataEC50:  200nMAssay Description:Effective concentration for half maximal stimulation of PI hydrolysis (mGluR1a)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM66976(SMR001230688 | trans-( )-ACPD monohydrate | cid_16...)
Affinity DataEC50:  2.20E+4nMAssay Description:Effective concentration for half maximal stimulation of PI hydrolysis (mGluR1a)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50053585((S)-4-(amino(carboxy)methyl)-2-hydroxybenzoic acid...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory concentration for half maximal inhibition of PI hydrolysis (mGluR1a)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50053588(4-((S)-Amino-carboxy-methyl)-benzoic acid | CHEMBL...)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibitory concentration for half maximal inhibition of PI hydrolysis (mGluR1a)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50030627(CHEMBL299683 | MCPG | (R,S)-alpha-Methyl-4-carboxy...)
Affinity DataIC50: 1.55E+5nMAssay Description:Inhibitory concentration for half maximal inhibition of PI hydrolysis (mGluR1a)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50030630(AIDA | AIDC | 1-Amino-indan-1,5-dicarboxylic acid(...)
Affinity DataIC50: 2.14E+5nMAssay Description:Inhibitory concentration for half maximal inhibition of PI hydrolysis (mGluR1a)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50053586(3C4HPG | CHEMBL128772 | 5-((S)-Amino-carboxy-methy...)
Affinity DataIC50: 2.90E+5nMAssay Description:Inhibitory concentration for half maximal inhibition of PI hydrolysis (mGluR1a)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed