Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 5047
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50005836(4-amino-5-chloro-N-(1-(3-(4-fluorophenoxy)propyl)-...)
Affinity DataKi:  25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82422(NSC_3035240 | CAS_109872-41-5 | RENZAPRIDE)
Affinity DataKi:  27nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82087(tryptamine, 5-Methoxy | 5-Methoxytryptamine hydroc...)
Affinity DataKi:  112nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50005836(4-amino-5-chloro-N-(1-(3-(4-fluorophenoxy)propyl)-...)
Affinity DataKi:  122nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  136nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  145nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50007871(CHEMBL8197 | ICS 205-930 | TROPISETRON)
Affinity DataKi:  159nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82422(NSC_3035240 | CAS_109872-41-5 | RENZAPRIDE)
Affinity DataKi:  243nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM81781(5-HT,omega-N-Me | 5-HT,a-Me)
Affinity DataKi:  263nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82087(tryptamine, 5-Methoxy | 5-Methoxytryptamine hydroc...)
Affinity DataKi:  401nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50007871(CHEMBL8197 | ICS 205-930 | TROPISETRON)
Affinity DataKi:  544nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  808nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM21392([3H]-5-carboxamidotryptamine | CHEMBL18840 | 5-car...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM81781(5-HT,omega-N-Me | 5-HT,a-Me)
Affinity DataKi:  1.45E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed