Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50003437
TargetBeta-2 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470923(CHEMBL122757)
Affinity DataKi:  0.302nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470917(CHEMBL120278)
Affinity DataKi:  1.5nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470918(CHEMBL123596)
Affinity DataKi:  1.5nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470916(CHEMBL121704)
Affinity DataKi:  2nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  2nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470924(CHEMBL122990)
Affinity DataKi:  6.5nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470919(CHEMBL332964)
Affinity DataKi:  7.80nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470922(CHEMBL122992)
Affinity DataKi:  8.70nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470920(CHEMBL121964)
Affinity DataKi:  12nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  44nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  47nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  79nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  79.4nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  162nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470923(CHEMBL122757)
Affinity DataKi:  178nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470923(CHEMBL122757)
Affinity DataKi:  182nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470918(CHEMBL123596)
Affinity DataKi:  186nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  324nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470922(CHEMBL122992)
Affinity DataKi:  355nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470924(CHEMBL122990)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470919(CHEMBL332964)
Affinity DataKi:  1.48E+3nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470921(CHEMBL333438)
Affinity DataKi:  4.37E+3nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470916(CHEMBL121704)
Affinity DataKi:  5.37E+3nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470920(CHEMBL121964)
Affinity DataKi:  1.91E+4nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470917(CHEMBL120278)
Affinity DataKi:  6.03E+4nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470921(CHEMBL333438)
Affinity DataKi:  8.32E+4nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed