Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50036431
TargetType-1 angiotensin II receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50236697(L-alpha-aspartyl-L-arginyl-L-valyl-L-tyrosyl-L-iso...)
Affinity DataKd:  2nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50052104(Sar-Arg-Val-Tyr-Asp-His-Apt-Phe | CHEMBL410812)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50052103(Sar-Arg-Val-Tyr-Glu-His-Apt-Phe | CHEMBL217873)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50052105(Sar-Arg-Val-Tyr-Cys-His-Pen-Phe | CHEMBL405938)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50052106(Sar-Arg-Val-Tyr-Cys-His-Mpc-Phe | CHEMBL406170)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50052108(Sar-Arg-Val-Tyr-Hcy-His-Mpc-Phe | CHEMBL415025)
Affinity DataKd:  20nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50052101(2-({1-[2-{2-[2-{2-[5-Guanidino-2-(2-methylamino-ac...)
Affinity DataKd:  0.540nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50052109(Sar-Arg-Val-Tyr-Cys-His-Mpt-Phe | CHEMBL412864)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50052102(Sar-Arg-Val-D-Tyr-Pro-His-Pro-Phe | CHEMBL414918)
Affinity DataKd:  58nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50052110(Sar-Arg-Val-Tyr-Hcy-His-Mpt-Phe | CHEMBL216678)
Affinity DataKd:  750nMAssay Description:Binding affinity was determined against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed