Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50006643
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50019293(cid_16362 | 1-(1-{3-[Bis-(4-fluoro-phenyl)-amino]-...)
Affinity DataIC50: 340nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50017702(cid_6365505 | 1-(bis(4-fluorophenyl)methyl)-4-cinn...)
Affinity DataIC50: 490nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051985(N-[3-(4-Benzyl-piperidin-1-yl)-propyl]-2,2-dipheny...)
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051984(N-[3-(4-Benzyl-piperazin-1-yl)-propyl]-2,2-dipheny...)
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051979(N-{3-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-pip...)
Affinity DataIC50: 720nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051978(2,2-Diphenyl-N-[3-(4-phenyl-piperidin-1-yl)-propyl...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051972(N-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051968(N-[3-(Benzyl-methyl-amino)-propyl]-2,2-diphenyl-ac...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051973(N-[3-(4-Phenoxy-piperidin-1-yl)-propyl]-2,2-diphen...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051976(N-[2-Methyl-3-(4-phenyl-piperidin-1-yl)-propyl]-2,...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051988(N-[3-(4-Hydroxy-4-phenyl-piperidin-1-yl)-propyl]-2...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051975(N-[3-(2,6-Dimethyl-morpholin-4-yl)-propyl]-2,2-dip...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043993(N-[3-(2,6-Dimethyl-piperidin-1-yl)-propyl]-2,2-dip...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051986(N-(3-Diethylamino-propyl)-2,2-diphenyl-acetamide |...)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051990(N-[3-(2,5-Dimethyl-pyrrolidin-1-yl)-propyl]-2,2-di...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051980(2,2-Diphenyl-N-(3-piperidin-1-yl-propyl)-acetamide...)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051982(N-(3-Morpholin-4-yl-propyl)-2,2-diphenyl-acetamide...)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051977(2,2-Diphenyl-N-(2-piperidin-1-yl-ethyl)-acetamide ...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051981(2,2-Diphenyl-N-(4-piperidin-1-yl-butyl)-acetamide ...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051987(N-(3-Dimethylamino-propyl)-2,2-diphenyl-acetamide ...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051983(N-[2-(1-Methyl-pyrrolidin-2-yl)-ethyl]-2,2-dipheny...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051974(N-(3-Amino-propyl)-2,2-diphenyl-acetamide | CHEMBL...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051989(N-(1-Aza-bicyclo[2.2.2]oct-3-yl)-2,2-diphenyl-acet...)
Affinity DataIC50: 9.50E+4nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051970(N-(3-Dimethylamino-propyl)-N-methyl-2,2-diphenyl-a...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50051969(N-[3-(4-Methyl-piperazin-1-yl)-propyl]-2,2-dipheny...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed